SCHEMBL5800641

SCHEMBL5800641

Cc1oc(-c2cccs2)nc1CC=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.50
ALDH1A1 P00352 8/20 0.50
HPGD P15428 6/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
NPSR1 Q6W5P4 2/20 0.50
POLB P06746 1/20 0.50
HSD17B10 Q99714 4/20 0.48
MAPT P10636 6/20 0.47
LMNA P02545 1/20 0.47
PPARA Q07869 5/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
PPARG P37231 4/20 0.44
PPARD Q03181 3/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP3A4 P08684 1/20 0.44
NPC1 O15118 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4748231 0.83 PPARA (0.64) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL13633793 0.82 KDM4E (0.54) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL4028821 0.81 KDM4E (0.53) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL1051606 0.81 KDM4E (0.53) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL12522017 0.81 KDM4E (0.53) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL13633782 0.79 HSD17B10 (0.53) KDM4EALDH1A1HPGDMEN1KMT2A
2-Thiophenenecarboxaldehyde SCHEMBL3976242 0.79 KDM4E (0.47) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL5098263 0.79 KDM4E (0.63) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL5228001 0.78 ALDH1A1 (0.52) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL7724076 0.78 KDM4E (0.51) KDM4EALDH1A1HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006057503-A1 NOVEL COMPOUNDS AS AGONIST FOR PPARϜ AND PPARα, METHOD FOR PREPARATION OF THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME LG LIFE SCIENCES, LTD. (KR) 2006-06-01 WO disclosed