SCHEMBL5801014

SCHEMBL5801014

C1=CN(c2cccc(-c3ccccc3)c2)c2ccccc2C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.41
HTR7 P34969 1/20 0.41
ALDH1A1 P00352 4/20 0.39
FAAH O00519 1/20 0.39
HSP90AA1 P07900 1/20 0.39
PKM P14618 1/20 0.39
HTT P42858 1/20 0.39
ATM Q13315 1/20 0.39
MGLL Q99685 1/20 0.39
COMT P21964 7/20 0.36
USP2 O75604 5/20 0.36
HSD17B10 Q99714 5/20 0.36
CYP1A2 P05177 4/20 0.36
CYP2D6 P10635 4/20 0.36
MAPK1 P28482 4/20 0.36
TP53 P04637 3/20 0.36
HIF1A Q16665 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
CYP3A4 P08684 2/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28286321 0.85 HPGD (0.39) ALDH1A1PKMUSP2SMN1; SMN2HPGD
SCHEMBL4148701 0.83 HPGD (0.38) ALDH1A1SMN1; SMN2HPGD
SCHEMBL4071380 0.83 HPGD (0.38) ALDH1A1SMN1; SMN2HPGD
SCHEMBL6578601 0.70 HSD17B3 (0.35) ALDH1A1CYP1A2CYP2D6HIF1ACYP3A4
SCHEMBL26058299 0.68 ALDH1A1 (0.48) HTR1AHTR7ALDH1A1FAAHHSP90AA1
SCHEMBL5572755 0.68 ALDH1A1 (0.34) ALDH1A1TSHR
SCHEMBL6576570 0.67 SLC6A4 (0.36) HTR1A
SCHEMBL5350419 0.66 PTGER1 (0.37) HTR1AHTR7ALDH1A1FAAHHSP90AA1
SCHEMBL6649618 0.65 PTGER1 (0.36) HTR1AHTR7ALDH1A1FAAHHSP90AA1
SCHEMBL181031 0.65 GRIN1 (0.41) ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1635829-A1 8-(3-BIARYL)PHENYLQUINOLINE PHOSPHODIESTERASE-4-INHIBITORS Merck Frosst Canada Ltd. (CA) 2006-03-22 EP disclosed
WO-2004096220-A1 8-(3-BIARYL)PHENYLQUINOLINE PHOSPHODIESTERASE-4-INHIBITORS MERCK FROSST CANADA LTD. (CA) 2004-11-11 WO disclosed