SCHEMBL5801185

SCHEMBL5801185

COC(=O)CC(N)c1ccc(NC(=O)c2c(Cl)cccc2Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.50
TAS1R3 Q7RTX0 2/20 0.48
TAS1R1 Q7RTX1 2/20 0.48
TAS1R2 Q8TE23 1/20 0.48
TYK2 P29597 4/20 0.48
JAK1 P23458 3/20 0.48
JAK2 O60674 3/20 0.48
CYP3A4 P08684 1/20 0.48
ITGB1 P05556 11/20 0.45
ITGA4 P13612 11/20 0.45
ITGA2 P17301 1/20 0.45
ITGB7 P26010 1/20 0.45
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5259497 0.88 ITGB1 (0.49) ITGB1ITGA4
SCHEMBL6511921 0.86 KMT2A (0.53) KMT2ATAS1R3TAS1R1TAS1R2TYK2
Trifluoroacetic Acid SCHEMBL6518249 0.81 ITGB1 (0.48) ITGB1ITGA4
SCHEMBL5257953 0.78 ITGB1 (0.47) ITGB1ITGA4
SCHEMBL3658423 0.76 L3MBTL1 (0.46) KMT2ACYP3A4MAPTRAB9A
SCHEMBL1294954 0.76 L3MBTL1 (0.46) KMT2ACYP3A4MAPTRAB9A
SCHEMBL391130 0.76 L3MBTL1 (0.46) KMT2ACYP3A4MAPTRAB9A
SCHEMBL28097862 0.75 JAK2 (0.51) KMT2ATAS1R3TAS1R1TAS1R2TYK2
Hydrochloric Acid SCHEMBL391129 0.75 L3MBTL1 (0.44) KMT2ACYP3A4MAPTRAB9A
Hydrochloric Acid SCHEMBL389435 0.75 L3MBTL1 (0.44) KMT2ACYP3A4MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006052962-A2 BICYCLIC TRIAZOLE A4 INTEGRIN INHIBITORS JANSSEN PHARMACEUTICA, N.V. (BE) 2006-05-18 WO disclosed