SCHEMBL5801661

SCHEMBL5801661

Cc1ccc(C(C)c2c[nH]cn2)cc1C

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.32
TRPA1 O75762 1/20 0.31
PTGS1 P23219 1/20 0.31
CACNA1C Q13936 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30673980 0.82 CHEK2 (0.35) TRPA1PTGS1CACNA1C
SCHEMBL21624997 0.82 CHEK2 (0.35) TRPA1PTGS1CACNA1C
SCHEMBL7251725 0.76 SMN1; SMN2 (0.38) LMNA
SCHEMBL10550330 0.75 LMNA (0.31) LMNATRPA1
SCHEMBL2104149 0.75 HTR2C (0.39) LMNA
SCHEMBL3753050 0.75 PTGS1 (0.47) PTGS1
SCHEMBL2104696 0.74 CYP19A1 (0.37)
SCHEMBL13256930 0.74 CYP3A4 (0.35)
SCHEMBL2336888 0.73 LMNA (0.46) LMNATRPA1PTGS1CACNA1C
SCHEMBL29352459 0.73 LMNA (0.46) LMNATRPA1PTGS1CACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663207-A2 NOVEL METHODS FOR IDENTIFYING IMPROVED, NON-SEDATING a-2 AGON ISTS Allergan, Inc. (US) 2006-06-07 EP disclosed
WO-2005034849-A2 METHODS FOR IDENTIFYING IMPROVED, NON-SEDATING ALPHA-2 AGONISTS ALLERGAN, INC. (US) 2005-04-21 WO disclosed