SCHEMBL5801700

SCHEMBL5801700

Cc1cc(C)cc(C(Br)C=O)c1

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.38
ALDH1A1 P00352 2/20 0.32
TSHR P16473 2/20 0.32
TPMT P51580 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4960285 0.79 ACP3 (0.43) ALDH1A1TSHR
SCHEMBL21597319 0.76 CYP2A6 (0.42) ALDH1A1
SCHEMBL2468299 0.76 CYP2A6 (0.42) ALDH1A1
SCHEMBL27961318 0.76 ERN1 (0.34) ERN1
SCHEMBL22833975 0.74 ERN1 (0.32) ERN1ALDH1A1
SCHEMBL3410995 0.74 ERN1 (0.32) ERN1ALDH1A1
SCHEMBL1100811 0.73 ERN1 (0.39) ERN1ALDH1A1TSHRTPMT
SCHEMBL15687876 0.71 BACE1 (0.38) TSHR
SCHEMBL21724409 0.71 TSHR (0.38) ERN1TSHRTPMT
SCHEMBL4709591 0.71 CES2 (0.38) ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3322705-A1 2-AMINO-1,3,4-THIADIAZINE AND 2-AMINO-1,3,4-OXADIAZINE BASED ANTIFUNGAL AGENTS F2G Limited (GB) 2018-05-23 EP disclosed
WO-2017009651-A1 2-AMINO-1,3,4-THIADIAZINE AND 2-AMINO-1,3,4-OXADIAZINE BASED ANTIFUNGAL AGENTS F2G LIMITED (GB) 2017-01-19 WO disclosed
EP-2822928-A1 SUBSTITUTED HETEROCYCLIC ACETAMIDES AS KAPPA OPIOID RECEPTOR (KOR) AGONISTS Dr. Reddy's Laboratories Ltd. (IN) 2015-01-14 EP disclosed
WO-2013131408-A1 SUBSTITUTED HETEROCYCLIC ACETAMIDES AS KAPPA OPIOID RECEPTOR (KOR) AGONISTS DR.REDDY'S LABORATORIES LTD. (IN) 2013-09-12 WO disclosed
WO-2006057503-A1 NOVEL COMPOUNDS AS AGONIST FOR PPARϜ AND PPARα, METHOD FOR PREPARATION OF THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME LG LIFE SCIENCES, LTD. (KR) 2006-06-01 WO disclosed