SCHEMBL21724409

SCHEMBL21724409

O=C[C@@H](Br)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.38
ERN1 O75460 3/20 0.38
TPMT P51580 1/20 0.31
TP53 P04637 1/20 0.31
CYP3A4 P08684 1/20 0.31
IDO1 P14902 1/20 0.31
TDO2 P48775 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1852012 0.86 ERN1 (0.32) ERN1
SCHEMBL169020 0.79 ACP3 (0.43) TSHR
SCHEMBL10350505 0.77 S1PR2 (0.33)
SCHEMBL1920603 0.77 HCAR2 (0.37)
SCHEMBL5725302 0.76 TSHR (0.38) TSHRTP53CYP3A4IDO1TDO2
SCHEMBL118609 0.76 HSD17B10 (0.42) TSHRTP53IDO1TDO2
SCHEMBL3979239 0.76 ERN1 (0.39) TSHRERN1CYP3A4
SCHEMBL4009249 0.76 ALDH1A1 (0.41) TSHRCYP3A4
SCHEMBL17431765 0.75 TSHR (0.42) TSHRERN1TPMTTP53CYP3A4
SCHEMBL3402042 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3836919-A1 1,3,4,9-TETRAHYDRO-2H-PYRIDO[3,4-B]INDOLE DERIVATIVE COMPOUNDS AND USES THEREOF Recreo Pharmaceuticals Inc. (US) 2021-06-23 EP disclosed
WO-2020037155-A1 1,3,4,9-TETRAHYDRO-2H-PYRIDO[3,4-B]INDOLE DERIVATIVE COMPOUNDS AND USES THEREOF RECREO PHARMACEUTICALS LLC (US) 2020-02-20 WO disclosed