SCHEMBL5801910

SCHEMBL5801910

COc1ccc2c(c1)c1c(n2CC(=O)O)-c2ccccc2NC(=O)C1

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 10/20 0.66
GSK3B P49841 11/20 0.58
CCNB2 O95067 9/20 0.58
CCNB1 P14635 9/20 0.58
CCNB3 Q8WWL7 9/20 0.58
CDK5 Q00535 1/20 0.53
CDK5R1 Q15078 1/20 0.53
AKR1B10 O60218 2/20 0.52
AKR1B1 P15121 2/20 0.52
AKR1A1 P14550 1/20 0.52
PTGDR2 Q9Y5Y4 3/20 0.48
GSK3A P49840 2/20 0.43
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
MDH2 P40926 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5801923 0.85 CDK1 (0.79) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5804773 0.82 CDK1 (0.58) CDK1GSK3BCCNB2CCNB1CCNB3
Hydrochloric Acid SCHEMBL5803457 0.82 CDK1 (0.57) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5818474 0.80 CDK1 (0.55) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5688713 0.80 CDK1 (1.00) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5803817 0.77 CDK1 (0.64) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5815923 0.75 CDK1 (0.56) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL6012263 0.73 GSK3B (1.00) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5805246 0.72 CDK1 (0.73) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL261494 0.72 CDK1 (0.48) CDK1GSK3BCCNB2CCNB1CCNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006089874-A1 BENZO[2,3]AZEPINO[4,5-B]INDOL-6-ONES GPC BIOTECH AG (DE) 2006-08-31 WO claimed
WO-2006089874-A1 BENZO[2,3]AZEPINO[4,5-B]INDOL-6-ONES GPC BIOTECH AG (DE) 2006-08-31 WO disclosed