SCHEMBL5804773

SCHEMBL5804773

O=C(O)Cn1c2c(c3cc(C(F)(F)F)ccc31)CC(=O)Nc1ccccc1-2

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 12/20 0.58
GSK3B P49841 14/20 0.56
CCNB2 O95067 11/20 0.56
CCNB1 P14635 11/20 0.56
CCNB3 Q8WWL7 11/20 0.56
CDK5 Q00535 5/20 0.53
CDK5R1 Q15078 5/20 0.53
PTGDR2 Q9Y5Y4 3/20 0.48
PTGDR Q13258 1/20 0.45
GSK3A P49840 3/20 0.42
AKR1B10 O60218 2/20 0.42
AKR1B1 P15121 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5801923 0.85 CDK1 (0.79) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5815923 0.84 CDK1 (0.56) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5802551 0.83 CDK1 (0.51) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5801910 0.82 CDK1 (0.66) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5802955 0.82 CDK1 (0.53) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5688713 0.74 CDK1 (1.00) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5688439 0.71 GSK3B (1.00) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL30319745 0.71 GSK3B (1.00) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL6012263 0.71 GSK3B (1.00) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5690667 0.71 GSK3B (0.78) CDK1GSK3BCCNB2CCNB1CCNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006089874-A1 BENZO[2,3]AZEPINO[4,5-B]INDOL-6-ONES GPC BIOTECH AG (DE) 2006-08-31 WO disclosed