SCHEMBL5815923

SCHEMBL5815923

COc1cc2c(cc1OC)-c1c(c3cc(C(F)(F)F)ccc3n1CC(=O)O)CC(=O)N2

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 10/20 0.56
CCNB2 O95067 9/20 0.56
CCNB1 P14635 9/20 0.56
GSK3B P49841 9/20 0.56
CCNB3 Q8WWL7 9/20 0.56
CDK5 Q00535 6/20 0.56
CDK5R1 Q15078 6/20 0.56
PTGDR2 Q9Y5Y4 7/20 0.41
PLK1 P53350 1/20 0.40
AKR1B1 P15121 2/20 0.39
AKR1B10 O60218 1/20 0.39
PTGDR Q13258 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5803817 0.86 CDK1 (0.64) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5819216 0.84 CDK1 (0.47) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5804773 0.84 CDK1 (0.58) CDK1CCNB2CCNB1GSK3BCCNB3
Hydrochloric Acid SCHEMBL5813979 0.84 CDK1 (0.47) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5802944 0.82 CDK1 (0.46) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5805683 0.76 CDK1 (0.65) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5801910 0.75 CDK1 (0.66) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5823198 0.73 CDK1 (0.57) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL5688837 0.72 GSK3B (1.00) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL30319820 0.72 GSK3B (1.00) CDK1CCNB2CCNB1GSK3BCCNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006089874-A1 BENZO[2,3]AZEPINO[4,5-B]INDOL-6-ONES GPC BIOTECH AG (DE) 2006-08-31 WO disclosed