SCHEMBL5804872

SCHEMBL5804872

COc1ccc(-c2[nH]c(C(C)C)c(C(=O)Nc3ccccc3)c2-c2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.46
KMT2A Q03164 4/20 0.46
POLB P06746 3/20 0.46
CTDSP1 Q9GZU7 2/20 0.46
GAA P10253 2/20 0.46
NPC1 O15118 3/20 0.46
ADORA3 P0DMS8 1/20 0.46
GSK3B P49841 2/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
KDM4E B2RXH2 1/20 0.44
CNR1 P21554 1/20 0.44
MEN1 O00255 3/20 0.43
ALDH1A1 P00352 1/20 0.43
HTT P42858 1/20 0.43
TRPV1 Q8NER1 1/20 0.43
KCNK9 Q9NPC2 1/20 0.43
AURKA O14965 1/20 0.42
PRKDC P78527 1/20 0.42
ATR Q13535 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5805083 0.91 EGFR (0.47) KMT2APOLBGAASMN1; SMN2MEN1
SCHEMBL4169210 0.86 HMGCR (0.47) RAB9AKMT2APOLBGAANPC1
SCHEMBL5804950 0.86 KDR (0.42) GAASMN1; SMN2
SCHEMBL5807727 0.85 HMGCR (0.46) RAB9AKMT2APOLBGAANPC1
SCHEMBL5808355 0.84 KCNK9 (0.43) RAB9AGAANPC1SMN1; SMN2KDM4E
SCHEMBL5804849 0.84 SLCO1B1 (0.45) RAB9AKMT2APOLBNPC1SMN1; SMN2
SCHEMBL5808861 0.84 HTT (0.45) POLBSMN1; SMN2ALDH1A1HTT
SCHEMBL5805311 0.84 HTT (0.45) POLBSMN1; SMN2ALDH1A1HTT
SCHEMBL5809279 0.83 MAPT (0.49) RAB9AKMT2APOLBGAANPC1
SCHEMBL5806885 0.81 CHEK1 (0.42) RAB9ANPC1SMN1; SMN2KDM4ECNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006110918-A1 PYRROLE COMPOUNDS AND USES THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2006-10-19 WO claimed
US-7323490-B2 Pyrrole compounds and uses thereof AMBIT BIOSCIENCES CORPORATION (US) 2008-01-29 US disclosed
WO-2006110918-A1 PYRROLE COMPOUNDS AND USES THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2006-10-19 WO disclosed