SCHEMBL5808355

SCHEMBL5808355

CC(C)c1[nH]c(-c2ccc(C(C)(C)C)cc2)c(-c2ccccc2)c1C(=O)Nc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNK9 Q9NPC2 1/20 0.43
CHEK1 O14757 2/20 0.41
EGFR P00533 2/20 0.41
KDR P35968 2/20 0.41
NR1H4 Q96RI1 1/20 0.41
TRPV1 Q8NER1 2/20 0.41
CNR1 P21554 1/20 0.41
MAPT P10636 3/20 0.40
UBE2N P61088 1/20 0.40
NPSR1 Q6W5P4 2/20 0.40
PTGS2 P35354 1/20 0.40
GAA P10253 1/20 0.40
RAB9A P51151 1/20 0.40
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GRIN2C Q14957 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5805083 0.91 EGFR (0.47) CHEK1EGFRKDRMAPTUBE2N
SCHEMBL5804950 0.86 KDR (0.42) CHEK1EGFRKDRNR1H4MAPT
SCHEMBL4169210 0.86 HMGCR (0.47) CHEK1EGFRKDRNR1H4MAPT
SCHEMBL5807727 0.85 HMGCR (0.46) CHEK1EGFRKDRNR1H4MAPT
SCHEMBL5804872 0.84 RAB9A (0.46) KCNK9TRPV1CNR1GAARAB9A
SCHEMBL5805311 0.84 HTT (0.45) CHEK1EGFRKDRMAPTUBE2N
SCHEMBL5808861 0.84 HTT (0.45) CHEK1EGFRKDRMAPTUBE2N
SCHEMBL5809279 0.83 MAPT (0.49) CHEK1EGFRKDRMAPTUBE2N
SCHEMBL5806885 0.81 CHEK1 (0.42) CHEK1EGFRKDRCNR1MAPT
SCHEMBL5806553 0.81 HMGCR (0.43) CHEK1EGFRKDRNR1H4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006110918-A1 PYRROLE COMPOUNDS AND USES THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2006-10-19 WO claimed
US-7323490-B2 Pyrrole compounds and uses thereof AMBIT BIOSCIENCES CORPORATION (US) 2008-01-29 US disclosed
WO-2006110918-A1 PYRROLE COMPOUNDS AND USES THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2006-10-19 WO disclosed