SCHEMBL5809279

SCHEMBL5809279

CC(C)c1[nH]c(-c2ccc(C#N)cc2)c(-c2ccccc2)c1C(=O)Nc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.49
UBE2N P61088 1/20 0.49
ALDH1A1 P00352 6/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
NPSR1 Q6W5P4 2/20 0.43
PPARG P37231 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
NR2E3 Q9Y5X4 1/20 0.43
NCOR2 Q9Y618 1/20 0.43
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43
TAS1R2 Q8TE23 1/20 0.43
KDM4E B2RXH2 3/20 0.42
HPGD P15428 3/20 0.42
GAA P10253 1/20 0.42
ATR Q13535 1/20 0.41
EGFR P00533 4/20 0.41
KDR P35968 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5805083 0.90 EGFR (0.47) MAPTUBE2NMEN1KMT2ATDP1
SCHEMBL5804950 0.85 KDR (0.42) MAPTUBE2NGAAEGFRKDR
SCHEMBL4169210 0.85 HMGCR (0.47) MAPTUBE2NMEN1KMT2AKDM4E
SCHEMBL5807727 0.84 HMGCR (0.46) MAPTUBE2NMEN1KMT2AKDM4E
SCHEMBL5804872 0.83 RAB9A (0.46) ALDH1A1MEN1KMT2AKDM4EGAA
SCHEMBL5808355 0.83 KCNK9 (0.43) MAPTUBE2NNPSR1KDM4EGAA
SCHEMBL5805311 0.83 HTT (0.45) MAPTUBE2NALDH1A1EGFRKDR
SCHEMBL5808861 0.83 HTT (0.45) MAPTUBE2NALDH1A1EGFRKDR
SCHEMBL5806885 0.80 CHEK1 (0.42) MAPTUBE2NALDH1A1KDM4EATR
SCHEMBL5806553 0.80 HMGCR (0.43) MAPTMEN1KMT2ANPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006110918-A1 PYRROLE COMPOUNDS AND USES THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2006-10-19 WO claimed
WO-2006110918-A1 PYRROLE COMPOUNDS AND USES THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2006-10-19 WO disclosed