SCHEMBL5807804

SCHEMBL5807804

COC(=O)C(c1ccccc1)C1(Cc2ccc(F)cc2)CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.48
TSHR P16473 2/20 0.44
ALOX15 P16050 1/20 0.44
P2RX7 Q99572 1/20 0.43
YAP1 P46937 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
TACR1 P25103 1/20 0.42
TP53 P04637 1/20 0.41
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 1/20 0.40
KDM4E B2RXH2 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
HDAC8 Q9BY41 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4036608 0.79 ATM (0.51) ATMTSHRALOX15P2RX7MEN1
SCHEMBL5671946 0.77 CNR1 (0.47) ATMTSHRALOX15MEN1KMT2A
SCHEMBL2792102 0.77 P2RX7 (0.52) ATMTSHRALOX15P2RX7YAP1
SCHEMBL23849296 0.77 TSHR (0.51) ATMTSHRALOX15TACR1KDM4E
SCHEMBL5674705 0.76 PKM (0.53) MEN1KMT2AHDAC1HDAC2CNR1
SCHEMBL2185224 0.76 KDM1A (0.46) ATMTSHRALOX15MEN1KMT2A
SCHEMBL4634595 0.76 KDM1A (0.46) ATMTSHRALOX15MEN1KMT2A
SCHEMBL14357682 0.76 KDM1A (0.48) ATMTSHRALOX15MEN1KMT2A
SCHEMBL5672765 0.76 KDM1A (0.48) ATMTSHRALOX15MEN1KMT2A
SCHEMBL4634695 0.76 HDAC2 (0.48) ATMTSHRALOX15MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006086609-A2 INHIBITORS OF TRYPTASE AXYS PHARMACEUTICALS, INC. (US) 2006-08-17 WO disclosed