SCHEMBL5808017

SCHEMBL5808017

COc1ccccc1OCC(=O)Nc1ccc2sc(C(=O)NO)cc2c1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 9/20 0.62
SMN1; SMN2 Q16637 2/20 0.56
MAPT P10636 4/20 0.55
NPC1 O15118 3/20 0.54
RAB9A P51151 2/20 0.54
POLB P06746 1/20 0.54
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
HPGD P15428 2/20 0.51
LMNA P02545 2/20 0.51
KDM4E B2RXH2 1/20 0.51
CDYL Q9Y232 1/20 0.51
TSHR P16473 1/20 0.50
NOTUM Q6P988 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5809353 0.85 HDAC1 (0.54) HDAC1MAPTLMNAKDM4E
SCHEMBL5809271 0.84 HDAC1 (0.71) HDAC1MAPTNPC1RAB9APOLB
SCHEMBL1890073 0.82 HDAC1 (0.67) HDAC1SMN1; SMN2MAPTPOLBHPGD
SCHEMBL6509116 0.79 HDAC1 (0.63) HDAC1
SCHEMBL5805563 0.79 HDAC1 (0.73) HDAC1
SCHEMBL1889466 0.78 HDAC1 (0.62) HDAC1
SCHEMBL12663159 0.77 HDAC1 (0.67) HDAC1SMN1; SMN2LMNAKDM4ETSHR
SCHEMBL1893680 0.77 HDAC1 (1.00) HDAC1
SCHEMBL1886036 0.77 HDAC1 (0.84) HDAC1SMN1; SMN2MAPTRAB9ALMNA
SCHEMBL8260320 0.77 HDAC1 (0.67) HDAC1SMN1; SMN2MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006101454-A1 BENZOTHIOPHENE DERIVATIVES: PREPARATION AND PHARMACEUTICAL APPLICATIONS S*BIO PTE LTD (SG) 2006-09-28 WO claimed