SCHEMBL5808501

SCHEMBL5808501

Cc1ccc(C(N)=O)c(C2CCNCC2)c1C

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.44
PARP1 P09874 11/20 0.42
CDC7 O00311 1/20 0.41
IKBKB O14920 1/20 0.38
CHUK O15111 1/20 0.38
PARP2 Q9UGN5 3/20 0.38
TLR9 Q9NR96 1/20 0.38
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
PLAT P00750 1/20 0.37
MEN1 O00255 1/20 0.36
CYP2D6 P10635 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3809365 0.82 PARP1 (0.51) HTR2CPARP1CDC7IKBKBCHUK
SCHEMBL28470220 0.82 MAPK1 (0.39) PARP1
SCHEMBL28325510 0.79 PARP1 (0.57) PARP1CDC7IKBKBCHUKPARP2
SCHEMBL28478841 0.77 F2 (0.38) PLAT
SCHEMBL2790537 0.76 ADRB1 (0.42) MEN1KMT2A
SCHEMBL30760594 0.76 QDPR (0.49) HTR2CPARP1CDC7IKBKBCHUK
SCHEMBL25436217 0.76 SIRT3 (0.37) PARP1MEN1CYP2D6KMT2A
SCHEMBL28571503 0.75 MKNK1 (0.46) PARP1PARP2
SCHEMBL28175941 0.74 MEN1 (0.43) PARP1CDC7MEN1KMT2A
SCHEMBL27544733 0.74 HTR2C (0.40) HTR2CPLATMEN1CYP2D6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615643-A1 4-PHENYL-PIPERIDINE COMPOUNDS AND THEIR USE AS MODULATORS OF OPIOID RECEPTORS Pfizer Products Inc. (US) 2006-01-18 EP disclosed
WO-2004089370-A1 4-PHENYL-PIPERIDINE COMPOUNDS AND THEIR USE AS MODULATORS OF OPIOID RECEPTORS PFIZER PRODUCTS INC. (US) 2004-10-21 WO disclosed