SCHEMBL580911

SCHEMBL580911

CCOC(=O)CC(=O)[C@@H]1CCN(C(=O)OC)[C@H](c2ccc(C(F)(F)F)cc2C)C1.COC(=O)N1CCC(C(=O)O)CC1c1ccc(C(F)(F)F)cc1C

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 9/20 0.40
ALDH1A1 P00352 2/20 0.38
NOTUM Q6P988 1/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
TMEM97 Q5BJF2 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
CETP P11597 1/20 0.35
MGLL Q99685 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL582517 0.96 TACR1 (0.42) TACR1ALDH1A1USP2LMNAMAPK1
SCHEMBL582518 0.96 TACR1 (0.42) TACR1ALDH1A1USP2LMNAMAPK1
SCHEMBL581119 0.90 NOTUM (0.43) TACR1NOTUMSIGMAR1
SCHEMBL599010 0.89 CYP11B1 (0.39) TACR1ALDH1A1USP2LMNAMAPK1
SCHEMBL581169 0.89 CYP11B1 (0.39) TACR1ALDH1A1USP2LMNAMAPK1
SCHEMBL581644 0.89 CYP11B1 (0.39) TACR1ALDH1A1USP2LMNAMAPK1
SCHEMBL581795 0.89 ALDH1A1 (0.47) ALDH1A1NOTUMUSP2LMNAMAPK1
SCHEMBL581796 0.89 ALDH1A1 (0.47) ALDH1A1NOTUMUSP2LMNAMAPK1
SCHEMBL581727 0.88 NOTUM (0.38) ALDH1A1NOTUMMAPK1
SCHEMBL581726 0.88 NOTUM (0.38) ALDH1A1NOTUMMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed