SCHEMBL581796

SCHEMBL581796

CCOC(=O)CC(=O)[C@@H]1CCN(C(=O)OC)[C@H](c2cccc(C(F)(F)F)c2)C1.COC(=O)N1CCC(C(=O)O)CC1c1cccc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
KCNN4 O15554 1/20 0.41
NOTUM Q6P988 1/20 0.40
KMT2A Q03164 2/20 0.39
LMNA P02545 2/20 0.39
USP2 O75604 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
CACNA1F O60840 1/20 0.39
CACNA1D Q01668 1/20 0.39
CACNA1S Q13698 1/20 0.39
CACNA1C Q13936 1/20 0.39
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
TRPV4 Q9HBA0 1/20 0.38
APOBEC3A P31941 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38
MEN1 O00255 1/20 0.37
HSP90AA1 P07900 1/20 0.37
ALOX15 P16050 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL581795 1.00 ALDH1A1 (0.47) ALDH1A1KCNN4NOTUMKMT2ALMNA
SCHEMBL3073129 0.96 ALDH1A1 (0.49) ALDH1A1KCNN4KMT2ALMNAUSP2
SCHEMBL580798 0.96 ALDH1A1 (0.49) ALDH1A1KCNN4KMT2ALMNAUSP2
SCHEMBL3062815 0.96 ALDH1A1 (0.49) ALDH1A1KCNN4KMT2ALMNAUSP2
SCHEMBL587487 0.92 ALDH1A1 (0.38) ALDH1A1KCNN4KMT2ATRPV4MEN1
SCHEMBL581727 0.89 NOTUM (0.38) ALDH1A1NOTUMMAPK1POLBSMN1; SMN2
SCHEMBL581726 0.89 NOTUM (0.38) ALDH1A1NOTUMMAPK1POLBSMN1; SMN2
SCHEMBL580827 0.89 NOTUM (0.48) ALDH1A1NOTUMKMT2ALMNAUSP2
SCHEMBL580911 0.89 TACR1 (0.40) ALDH1A1NOTUMLMNAUSP2MAPK1
SCHEMBL581242 0.88 ALDH1A1 (0.40) ALDH1A1KCNN4KMT2ATRPV4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed