SCHEMBL5809728

SCHEMBL5809728

CC(/C=C/C(=O)N1CCCC1)=C\c1ccc2c(c1)OCO2.CC(/C=C/C(=O)N1CCCCC1)=C\c1ccc2c(c1)OCO2.CCN(CC)C(=O)/C=C/C(C)=C/c1ccc2c(c1)OCO2

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 4/20 0.59
TRPV1 Q8NER1 3/20 0.59
NPC1 O15118 2/20 0.59
RAB9A P51151 2/20 0.59
MAOB P27338 4/20 0.57
KDM4E B2RXH2 5/20 0.56
ALDH1A1 P00352 5/20 0.56
HPGD P15428 5/20 0.56
CYP3A4 P08684 3/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
HSD17B10 Q99714 2/20 0.56
GABRA1 P14867 2/20 0.56
GABRB2 P47870 2/20 0.56
CTSD P07339 1/20 0.56
ABCB1 P08183 1/20 0.56
ALOX5 P09917 1/20 0.56
MAOA P21397 1/20 0.56
MAPK1 P28482 1/20 0.56
DHODH Q02127 1/20 0.56
HDAC6 Q9UBN7 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14597900 0.89 TRPV1 (0.73) TRPV1NPC1RAB9AMAOBKDM4E
SCHEMBL5494471 0.88 MAOB (0.72) TRPV1NPC1RAB9AMAOBKDM4E
SCHEMBL5494974 0.88 TRPM8 (0.74) TRPM8KDM4EALDH1A1HPGDCYP3A4
SCHEMBL5494975 0.88 TRPM8 (0.74) TRPM8KDM4EALDH1A1HPGDCYP3A4
SCHEMBL29359315 0.81 TRPV1 (0.67) TRPV1NPC1RAB9AMAOBKDM4E
SCHEMBL5494854 0.80 MAOB (0.66) TRPV1NPC1RAB9AMAOBKDM4E
SCHEMBL5496910 0.77 TRPM8 (0.71) TRPM8KDM4EALDH1A1HPGDCYP3A4
SCHEMBL5496911 0.77 TRPM8 (0.71) TRPM8KDM4EALDH1A1HPGDCYP3A4
SCHEMBL5493158 0.76 RAB9A (0.56) TRPV1NPC1RAB9AMAOBKDM4E
Ilepcimide SCHEMBL668328 0.75 NPC1 (1.00) TRPV1NPC1RAB9AMAOBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006103527-A1 AROMATIC SUBSTITUTED PENTADIENOIC ACID AMIDE FOR COMBINATION WITH ANTI-INFECTIVE DRUGS COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2006-10-05 WO disclosed