SCHEMBL5810372

SCHEMBL5810372

C#CCNc1nc2ccc(OC(F)(F)F)cc2n1CC#C

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPC5 Q9UL62 1/20 0.39
IDH1 O75874 11/20 0.38
PDE10A Q9Y233 2/20 0.38
PDE2A O00408 1/20 0.38
PDE7A Q13946 1/20 0.38
PDE11A Q9HCR9 1/20 0.38
BRD4 O60885 4/20 0.36
PPARG P37231 1/20 0.35
ACACB O00763 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5822557 0.99 TRPC5 (0.38) TRPC5IDH1PDE10APDE2APDE7A
SCHEMBL5806451 0.91 TRPC5 (0.45) TRPC5IDH1BRD4
Hydrochloric Acid SCHEMBL5810454 0.90 TRPC5 (0.44) TRPC5IDH1BRD4
Hydrochloric Acid SCHEMBL5806513 0.86 PPARG (0.42) IDH1PDE10APDE2APDE7APDE11A
Hydrochloric Acid SCHEMBL5809663 0.79 ALDH1A1 (0.48) TRPC5IDH1BRD4
SCHEMBL6250112 0.70 DYRK1A (0.61)
Hydrochloric Acid SCHEMBL6834656 0.69 DYRK1A (0.60)
SCHEMBL4233355 0.66 POLB (0.51)
SCHEMBL31020720 0.66 TRPV1 (0.41) TRPC5IDH1
SCHEMBL15730236 0.64 PPARG (0.45) IDH1PDE10APDE2APDE7APDE11A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006050148-A2 PROPARGYL TRIFLUOROMETHOXY AMINOBENZIMIDAZOLE DERIVATIVES TEVA PHARMACEUTICAL INDUSTRIES, LTD. (IL) 2006-05-11 WO disclosed