SCHEMBL5812504

SCHEMBL5812504

Fc1cc(C[CH]c2ccc3ccccc3c2)cc(F)c1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RELA Q04206 1/20 0.42
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAPT P10636 2/20 0.39
GLA P06280 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
RAB9A P51151 1/20 0.39
CYP1A2 P05177 2/20 0.38
CYP2A6 P11509 2/20 0.38
PTGS1 P23219 1/20 0.38
NQO2 P16083 2/20 0.36
GRIN2D O15399 2/20 0.35
GRIN3B O60391 2/20 0.35
GRIN1 Q05586 2/20 0.35
GRIN2A Q12879 2/20 0.35
GRIN2B Q13224 2/20 0.35
GRIN2C Q14957 2/20 0.35
GRIN3A Q8TCU5 2/20 0.35
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8668861 0.80 RAB9A (0.51) RELAALDH1A1KDM4EL3MBTL1MAPT
SCHEMBL8204171 0.80 RELA (0.53) RELAALDH1A1KDM4EL3MBTL1MAPT
SCHEMBL7220223 0.75 CYP1A2 (0.48) RELAALDH1A1KDM4EL3MBTL1RAB9A
SCHEMBL8667992 0.75 RELA (0.43) RELAALDH1A1KDM4EL3MBTL1MAPT
SCHEMBL28140562 0.72 RELA (0.52) RELAALDH1A1KDM4EL3MBTL1MAPT
SCHEMBL8668276 0.71 CYP2D6 (0.48) RELACYP1A2
SCHEMBL140015 0.70 RELA (0.54) RELAALDH1A1KDM4EL3MBTL1MAPT
SCHEMBL8598224 0.70 NQO2 (0.50) MAPTSMN1; SMN2CYP1A2CYP2A6NQO2
SCHEMBL8710672 0.69 CYP1A2 (0.50) RELARAB9ACYP1A2CYP2A6
SCHEMBL9527298 0.69 RELA (0.52) RELAALDH1A1KDM4EL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615890-A1 PIPERIDINE DERIVATIVES AS RENIN INHIBITORS FOR THE TREATMENT OF HYPERTENSION WARNER-LAMBERT COMPANY (US) 2006-01-18 EP disclosed
WO-2004089903-A1 PIPERIDINE DERIVATIVES AS RENIN INHIBITORS FOR THE TREATMENT OF HYPERTENSION WARNER-LAMBERT COMPANY LLC (US) 2004-10-21 WO disclosed