SCHEMBL5812965

SCHEMBL5812965

NC(=O)C#Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.45
RPS6KA3 P51812 1/20 0.42
JAK3 P52333 1/20 0.42
GAA P10253 1/20 0.41
RXRA P19793 3/20 0.37
RXRG P48443 3/20 0.37
RXRB P28702 2/20 0.37
MAPT P10636 1/20 0.37
ITGB3 P05106 1/20 0.37
ITGAV P06756 1/20 0.37
TAS2R14 Q9NYV8 1/20 0.36
GPR35 Q9HC97 1/20 0.34
P2RX1 P51575 3/20 0.34
LMNA P02545 1/20 0.34
FFAR1 O14842 1/20 0.34
PTPN1 P18031 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6653912 0.98 CES2 (0.44) CES2RPS6KA3JAK3GAARXRA
SCHEMBL20569584 0.84 P2RX1 (0.41) GAAMAPTP2RX1LMNA
SCHEMBL6553318 0.82 CES2 (0.47) CES2RPS6KA3JAK3RXRARXRG
SCHEMBL8024378 0.81 CES2 (0.45) CES2PTPN1
SCHEMBL6553779 0.77 NOTUM (0.41) CES2GAAMAPTTAS2R14GPR35
SCHEMBL26328057 0.72 TAS2R14 (0.40) CES2RXRARXRGRXRBMAPT
SCHEMBL16503534 0.69 CES2 (0.35) CES2MAPTTAS2R14
SCHEMBL7997120 0.69 TAS2R14 (0.47) CES2MAPTITGB3ITGAVTAS2R14
SCHEMBL5540303 0.69 CES2 (0.38) CES2RPS6KA3JAK3RXRARXRG
SCHEMBL627995 0.69 CES2 (0.67) CES2RPS6KA3JAK3GAARXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638935-A1 NK1 ANTAGONIST Pfizer Products Inc. (US) 2006-03-29 EP disclosed
WO-2004110996-A1 NK1 ANTAGONIST PFIZER PRODUCTS INC. (US) 2004-12-23 WO disclosed
EP-1472256-A1 PIPERIDINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2004-11-03 EP disclosed
WO-2003066635-A1 PIPERIDINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2003-08-14 WO disclosed