SCHEMBL5814243

SCHEMBL5814243

COc1ccc(CNc2nc(-c3ccno3)nc3sc(C)c(C)c23)cc1Cl.Cc1sc2nc(-c3ccno3)nc(Cl)c2c1C

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BCDIN3D Q7Z5W3 2/20 0.40
CHRM4 P08173 1/20 0.40
PDE5A O76074 9/20 0.40
GAA P10253 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
PRKCI P41743 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5120646 0.97 BCDIN3D (0.42) BCDIN3DCHRM4PDE5AGAARXFP1
SCHEMBL7513169 0.94 CHRM4 (0.40) CHRM4PDE5AGAARXFP1PRKCI
SCHEMBL7514448 0.92 BCDIN3D (0.40) BCDIN3DCHRM4PDE5A
SCHEMBL5809508 0.91 GAA (0.40) CHRM4GAARXFP1PRKCI
SCHEMBL5128434 0.90 BCDIN3D (0.42) BCDIN3DCHRM4PDE5A
SCHEMBL5127812 0.89 MEN1 (0.42) CHRM4GAARXFP1PRKCI
SCHEMBL5130870 0.87 GAA (0.42) CHRM4GAARXFP1PRKCI
SCHEMBL5812974 0.86 CHRM4 (0.40) BCDIN3DCHRM4PDE5AGAA
SCHEMBL5820926 0.85 ALDH1A1 (0.44) CHRM4PDE5AGAARXFP1PRKCI
SCHEMBL5813640 0.84 PRKCI (0.44) PRKCI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685136-A1 USE OF THIENOPYRIMIDINES MERCK PATENT GmbH (DE) 2006-08-02 EP disclosed
WO-2005047292-A1 USE OF THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2005-05-26 WO disclosed