SCHEMBL5812974

SCHEMBL5812974

COc1ccc(CNc2nc(-c3ccno3)nc3sc(C)c(Cl)c23)cc1OC.Cc1sc2nc(-c3ccno3)nc(Cl)c2c1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 1/20 0.40
TSHR P16473 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TNF P01375 1/20 0.37
NOD1 Q9Y239 1/20 0.37
BCHE P06276 2/20 0.36
ACHE P22303 2/20 0.36
STAT1 P42224 1/20 0.36
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
APP P05067 2/20 0.35
PDE5A O76074 1/20 0.35
GAA P10253 2/20 0.35
POLB P06746 1/20 0.35
EGFR P00533 1/20 0.35
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5116928 0.97 CHRM4 (0.42) CHRM4TSHRMEN1KMT2ATNF
SCHEMBL7514448 0.94 BCDIN3D (0.40) CHRM4PDE5ABCDIN3D
SCHEMBL7513169 0.92 CHRM4 (0.40) CHRM4TSHRMEN1KMT2ATNF
SCHEMBL5128434 0.91 BCDIN3D (0.42) CHRM4PDE5ABCDIN3D
SCHEMBL7516123 0.88 USP1 (0.34) CHRM4KMT2ALMNAGAADYRK1A
SCHEMBL5127812 0.88 MEN1 (0.42) CHRM4TSHRMEN1KMT2ATNF
SCHEMBL5814243 0.86 BCDIN3D (0.40) CHRM4PDE5AGAABCDIN3D
SCHEMBL5813871 0.85 MEN1 (0.46) CHRM4TSHRMEN1KMT2ATNF
SCHEMBL5814517 0.85 ESR1 (0.43) CHRM4TSHRMEN1KMT2ATNF
SCHEMBL5814655 0.84 CHRM4 (0.40) CHRM4MEN1KMT2ALMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685136-A1 USE OF THIENOPYRIMIDINES MERCK PATENT GmbH (DE) 2006-08-02 EP disclosed
WO-2005047292-A1 USE OF THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2005-05-26 WO disclosed
EP-0920431-A1 THIENOPYRIMIDINES MERCK PATENT GmbH (DE) 1999-06-09 EP disclosed
WO-1998006722-A1 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 1998-02-19 WO disclosed