SCHEMBL5814543

SCHEMBL5814543

CCCCCN1CCC2(CC1)CN(C(=O)c1ccccc1Cl)c1ccc(F)cc12

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.46
SLC18A3 Q16572 1/20 0.46
DRD2 P14416 5/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
AVPR2 P30518 1/20 0.40
GNRHR P30968 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5578618 0.97 SIGMAR1 (0.46) SIGMAR1SLC18A3DRD2AVPR2
SCHEMBL5578571 0.87 NOTUM (0.43) GNRHR
SCHEMBL5578889 0.87 SIGMAR1 (0.43) SIGMAR1DRD2
SCHEMBL5616199 0.87 SIGMAR1 (0.43) SIGMAR1SLC18A3DRD2
SCHEMBL5578880 0.84 KDM2B (0.42)
SCHEMBL5578766 0.84 HDAC1 (0.38) SIGMAR1SLC18A3GNRHR
SCHEMBL14366293 0.83 OPRM1 (0.45) SIGMAR1
SCHEMBL5578753 0.83 HDAC1 (0.47) SIGMAR1
SCHEMBL5616027 0.81 SIGMAR1 (0.43) SIGMAR1SLC18A3LMNA
SCHEMBL5578687 0.80 KMT2A (0.48) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716148-A2 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF Arena Pharmaceuticals, Inc. (US) 2006-11-02 EP disclosed
WO-2005063745-A2 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARMACEUTICALS, INC. (US) 2005-07-14 WO disclosed