SCHEMBL5814849

SCHEMBL5814849

O=C(O)n1cc(CBr)c2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
MAPT P10636 1/20 0.44
RECQL P46063 1/20 0.44
OXER1 Q8TDS5 1/20 0.43
KDM4E B2RXH2 3/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
FABP3 P05413 1/20 0.39
FABP4 P15090 1/20 0.39
FABP5 Q01469 1/20 0.39
CREBBP Q92793 1/20 0.38
CDC25A P30304 1/20 0.38
GLA P06280 1/20 0.38
PLK1 P53350 1/20 0.37
THRB P10828 1/20 0.37
KMT2A Q03164 1/20 0.37
GPR84 Q9NQS5 1/20 0.37
IL6ST P40189 1/20 0.37
BCHE P06276 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5992534 0.87 OXER1 (0.47) ALDH1A1MAPTRECQLOXER1KDM4E
SCHEMBL28033575 0.85 KMT2A (0.54) ALDH1A1OXER1KDM4EL3MBTL1THRB
SCHEMBL5742862 0.83 OXER1 (0.41) ALDH1A1MAPTRECQLOXER1KDM4E
SCHEMBL2467334 0.83 CDC25A (0.54) ALDH1A1OXER1KDM4EL3MBTL1AKR1C3
SCHEMBL10442568 0.80 OXER1 (0.56) OXER1KDM4EFABP3FABP4FABP5
SCHEMBL5304010 0.80 HTR2A (0.57) ALDH1A1MAPTRECQLOXER1
SCHEMBL18423465 0.80 ALDH1A1 (0.59) ALDH1A1MAPTRECQLOXER1L3MBTL1
SCHEMBL351754 0.80 ALDH1A1 (0.59) ALDH1A1MAPTRECQLOXER1L3MBTL1
SCHEMBL11895393 0.80 ALDH1A1 (0.59) ALDH1A1MAPTRECQLOXER1L3MBTL1
SCHEMBL4518718 0.79 STAT3 (0.42) ALDH1A1MAPTRECQLOXER1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020243135-A1 FUSED HETEROCYCLIC DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2020-12-03 WO disclosed
EP-2448939-B1 2,3-DIHYDRO-1H-IMIDAZO {1,2-A} PYRIMIDIN-5-ONE DERIVATIVES, THE PREPARATION AND PHARMACEUTICAL USE THEREOF SANOFI SA (FR) 2017-03-01 EP disclosed
WO-2006061126-A2 DIBENZOXAZEPINONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2006-06-15 WO disclosed