SCHEMBL28033575

SCHEMBL28033575

O=C(c1ccccc1)n1cc(CBr)c2ccccc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.54
KDM4E B2RXH2 2/20 0.54
ALDH1A1 P00352 1/20 0.54
THRB P10828 1/20 0.54
ALOX5 P09917 1/20 0.49
HTR6 P50406 3/20 0.48
HTR1A P08908 1/20 0.48
HTR1D P28221 1/20 0.48
HTR1B P28222 1/20 0.48
HTR1F P30939 1/20 0.48
HTR7 P34969 1/20 0.48
PTGS2 P35354 4/20 0.46
DYRK1A Q13627 1/20 0.46
TSHR P16473 1/20 0.45
RAB9A P51151 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
P2RX4 Q99571 1/20 0.45
MEN1 O00255 1/20 0.44
OXER1 Q8TDS5 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16072693 0.86 KMT2A (0.58) KMT2AKDM4EALDH1A1THRBALOX5
SCHEMBL5814849 0.85 ALDH1A1 (0.44) KMT2AKDM4EALDH1A1THRBL3MBTL1
SCHEMBL27487257 0.82 HTR2A (0.53) KMT2AKDM4EALDH1A1THRBALOX5
SCHEMBL9629984 0.82 KMT2A (0.51) KMT2AKDM4EALDH1A1THRBALOX5
SCHEMBL10696303 0.82 OXER1 (0.56) KMT2AKDM4EALDH1A1THRBALOX5
SCHEMBL5444461 0.80 OXER1 (0.64) KMT2AKDM4EALDH1A1THRBALOX5
SCHEMBL16038911 0.80 KMT2A (0.56) KMT2AKDM4EALDH1A1THRBALOX5
SCHEMBL13125600 0.79 KMT2A (0.47) KMT2AKDM4EALDH1A1THRBALOX5
SCHEMBL13125598 0.79 KMT2A (0.48) KMT2AKDM4EALDH1A1THRBALOX5
SCHEMBL24877919 0.79 HTR6 (0.76) KMT2AKDM4EALDH1A1THRBHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104876848-B 1-benzoyl-3-indolyl thioester compound and preparation method thereof 南开大学 2017-05-17 CN claimed
CN-104876848-A 1-benzoyl-3-indolyl thioester compound and preparation method thereof UNIV NANKAI 2015-09-02 CN claimed
CN-104876848-B 1-benzoyl-3-indolyl thioester compound and preparation method thereof 南开大学 2017-05-17 CN disclosed
CN-104876848-B 1-benzoyl-3-indolyl thioester compound and preparation method thereof 南开大学 2017-05-17 CN disclosed
CN-104876848-A 1-benzoyl-3-indolyl thioester compound and preparation method thereof UNIV NANKAI 2015-09-02 CN disclosed
CN-104876848-A 1-benzoyl-3-indolyl thioester compound and preparation method thereof UNIV NANKAI 2015-09-02 CN disclosed