SCHEMBL5815028

SCHEMBL5815028

CSc1nc(Nc2ccc(N3CCOCC3)cc2)cc(N2CCN(CC(=O)N3CCC(C)CC3)CC2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
NPC1 O15118 1/20 0.46
HSD17B10 Q99714 1/20 0.46
AURKA O14965 4/20 0.42
AURKB Q96GD4 2/20 0.42
CYP1A2 P05177 1/20 0.41
NAMPT P43490 1/20 0.41
RIPK1 Q13546 1/20 0.41
ZAP70 P43403 1/20 0.40
EPHX2 P34913 1/20 0.40
RET P07949 1/20 0.40
KDR P35968 4/20 0.39
BRAF P15056 2/20 0.39
RAF1 P04049 1/20 0.39
PDGFRB P09619 1/20 0.39
KIT P10721 1/20 0.39
FGFR1 P11362 1/20 0.39
TEK Q02763 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5820442 0.92 HRH3 (0.43) AURKAAURKBCYP1A2NAMPTRIPK1
SCHEMBL5820856 0.92 AURKA (0.41) RAB9AAURKAAURKBCYP1A2NAMPT
SCHEMBL5822993 0.91 AURKA (0.42) AURKAAURKBCYP1A2NAMPTRIPK1
SCHEMBL5820310 0.91 HRH3 (0.45) AURKAAURKBCYP1A2NAMPTRIPK1
SCHEMBL5821064 0.91 SMN1; SMN2 (0.44) RAB9AKMT2AMEN1NPC1HSD17B10
SCHEMBL5820813 0.91 NAMPT (0.47) RAB9AKMT2ANPC1AURKAAURKB
SCHEMBL5820251 0.91 CYP1A2 (0.45) RAB9AKMT2AMEN1NPC1AURKA
SCHEMBL5820606 0.91 KDM4E (0.44) RAB9ANPC1HSD17B10AURKAAURKB
SCHEMBL5823039 0.90 AURKA (0.50) RAB9AKMT2ANPC1AURKAAURKB
SCHEMBL5823980 0.90 ZAP70 (0.49) RAB9AKMT2ANPC1AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006137706-A1 6-(4-SUBSTITUTED-ANILINO)PYRIMIDINE DERIVATIVES, METHOD FOR PREPARING THEREOF AND ANTIVIRAL PHARMACEUTICAL COMPOSITION COMPRISING THE SAME B & C BIOPHARM. CO., LTD. (KR) 2006-12-28 WO claimed
WO-2006137706-A1 6-(4-SUBSTITUTED-ANILINO)PYRIMIDINE DERIVATIVES, METHOD FOR PREPARING THEREOF AND ANTIVIRAL PHARMACEUTICAL COMPOSITION COMPRISING THE SAME B & C BIOPHARM. CO., LTD. (KR) 2006-12-28 WO disclosed