SCHEMBL5822993

SCHEMBL5822993

CSc1nc(Nc2ccc(N3CCOCC3)cc2)cc(N2CCN(CC(=O)N3CCC(C(N)=O)CC3)CC2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 4/20 0.42
AURKB Q96GD4 2/20 0.42
RIPK1 Q13546 1/20 0.41
CYP1A2 P05177 1/20 0.40
NAMPT P43490 1/20 0.39
ZAP70 P43403 1/20 0.39
RET P07949 1/20 0.39
EPHX2 P34913 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
EML4 Q9HC35 1/20 0.38
ALK Q9UM73 1/20 0.38
PIK3CA P42336 2/20 0.38
MTOR P42345 2/20 0.38
PIK3CD O00329 1/20 0.38
PIK3CB P42338 1/20 0.38
KDR P35968 2/20 0.38
BRAF P15056 1/20 0.38
MAPK9 P45984 1/20 0.38
MAPK10 P53779 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5815028 0.91 RAB9A (0.46) AURKAAURKBRIPK1CYP1A2NAMPT
SCHEMBL5820442 0.90 HRH3 (0.43) AURKAAURKBRIPK1CYP1A2NAMPT
SCHEMBL5820856 0.90 AURKA (0.41) AURKAAURKBRIPK1CYP1A2NAMPT
SCHEMBL5820310 0.89 HRH3 (0.45) AURKAAURKBRIPK1CYP1A2NAMPT
SCHEMBL5820251 0.89 CYP1A2 (0.45) AURKAAURKBCYP1A2NAMPTZAP70
SCHEMBL5821064 0.89 SMN1; SMN2 (0.44) AURKAAURKBCYP1A2NAMPTZAP70
SCHEMBL5820813 0.89 NAMPT (0.47) AURKAAURKBCYP1A2NAMPTZAP70
SCHEMBL5820606 0.88 KDM4E (0.44) AURKAAURKBRIPK1CYP1A2NAMPT
SCHEMBL5823039 0.88 AURKA (0.50) AURKAAURKBCYP1A2NAMPTZAP70
SCHEMBL5823980 0.88 ZAP70 (0.49) AURKAAURKBCYP1A2NAMPTZAP70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006137706-A1 6-(4-SUBSTITUTED-ANILINO)PYRIMIDINE DERIVATIVES, METHOD FOR PREPARING THEREOF AND ANTIVIRAL PHARMACEUTICAL COMPOSITION COMPRISING THE SAME B & C BIOPHARM. CO., LTD. (KR) 2006-12-28 WO claimed