SCHEMBL5815988

SCHEMBL5815988

Nc1sc(CCNC(=O)O)nc1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.46
ALDH1A1 P00352 5/20 0.45
GAA P10253 3/20 0.45
POLB P06746 1/20 0.45
PDE10A Q9Y233 1/20 0.43
CYP1A2 P05177 2/20 0.43
HSD17B10 Q99714 2/20 0.41
MAPK1 P28482 2/20 0.40
NTRK1 P04629 1/20 0.40
MAPT P10636 4/20 0.39
LMNA P02545 2/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HSP90AB1 P08238 1/20 0.39
HIF1A Q16665 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PTGS2 P35354 1/20 0.38
TP53 P04637 1/20 0.38
THRB P10828 1/20 0.38
XIAP P98170 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5815983 0.72 CYP1A2 (0.43) ALDH1A1GAAPOLBCYP1A2HSD17B10
SCHEMBL27684678 0.72 ALDH1A1 (0.41) ALDH1A1GAAPOLBCYP1A2HSD17B10
SCHEMBL4141222 0.70 MAPT (0.40) BTKALDH1A1HSD17B10MAPK1MAPT
SCHEMBL1721531 0.70 CYP1A2 (0.46) ALDH1A1GAAPOLBCYP1A2HSD17B10
SCHEMBL21916304 0.68 MME (0.41) ALDH1A1GAAPOLBCYP1A2MAPT
SCHEMBL8557878 0.68 ALDH1A1 (0.63) ALDH1A1GAAPOLBCYP1A2HSD17B10
SCHEMBL4125428 0.67 MAPT (0.38) ALDH1A1GAAMAPTLMNAHIF1A
SCHEMBL544732 0.67 ALDH1A1 (0.62) ALDH1A1GAAPOLBCYP1A2HSD17B10
SCHEMBL544015 0.67 ALDH1A1 (0.77) ALDH1A1POLBCYP1A2HSD17B10MAPK1
SCHEMBL543809 0.67 NTRK1 (0.51) ALDH1A1GAAPOLBCYP1A2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006085815-A1 THIAZOLE DERIVATIVES, THEIR PROCESS FOR THEIR PREPARATION AND THEIR USE IN THERAPY ASTRAZENECA AB (SE) 2006-08-17 WO disclosed