SCHEMBL5817142

SCHEMBL5817142

[2H]c1[nH]c2ccc(OC)cc2c1C[CH2]

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 2/20 0.59
HTR2B P41595 4/20 0.56
HTR2A P28223 6/20 0.54
HTR1A P08908 5/20 0.54
HTR2C P28335 4/20 0.54
HTR1D P28221 3/20 0.54
HTR1B P28222 3/20 0.54
HTR7 P34969 3/20 0.54
HTR6 P50406 3/20 0.54
CYP2D6 P10635 2/20 0.54
CYP1A2 P05177 2/20 0.54
HTR4 Q13639 2/20 0.54
MAPT P10636 2/20 0.54
TSHR P16473 2/20 0.54
NFKB1 P19838 1/20 0.54
TRPM8 Q7Z2W7 1/20 0.54
BLM P54132 1/20 0.52
PMP22 Q01453 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
KDM4E B2RXH2 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL217937 0.85 GPR84 (0.76) GPR84HTR2BHTR2AHTR1AHTR2C
Mebufotenin SCHEMBL33563480 0.80 HTR2A (0.54) GPR84HTR2BHTR2AHTR1AHTR2C
Melatonin SCHEMBL5815299 0.76 MTNR1A (0.78) HTR2BHTR1AHTR2CCYP2D6CYP1A2
SCHEMBL5431365 0.75 GPR84 (1.00) GPR84HTR2BHTR2AHTR1AHTR2C
SCHEMBL16824132 0.74 SLC6A4 (0.71) GPR84HTR2BHTR2AHTR1AHTR2C
SCHEMBL178561 0.73 GPR84 (0.78) GPR84HTR2BHTR2AHTR1AHTR2C
SCHEMBL947733 0.72 GPR84 (0.76) GPR84HTR2BHTR2AHTR1AHTR2C
SCHEMBL1723383 0.72 CYP2D6 (0.77) GPR84HTR2BHTR2AHTR1AHTR2C
SCHEMBL3976318 0.72 HTR2B (1.00) GPR84HTR2BHTR2AHTR1AHTR2C
SCHEMBL2125628 0.72 HTR2A (0.68) GPR84HTR2BHTR2AHTR1AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006086978-A2 USE OF DEUTERATED N-[2-(5-METHOXY-1H-INDOL-3-YL)-ETHYL]ACETAMIDES AND THE PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, AND MEDICAMENTS CONTAINING SAID COMPOUNDS BIRDS PHARMA GMBH BEROLINA INNOVATIVE RESEARCH & DEVELOPMENT SERVICES (DE) 2006-08-24 WO claimed