SCHEMBL5818356

SCHEMBL5818356

CCN(c1ccccc1)c1nccc(-c2sc(C3(O)CCNCC3)nc2-c2cccc(F)c2)n1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 4/20 0.36
MAPKAPK2 P49137 1/20 0.34
BRAF P15056 3/20 0.33
KMO O15229 1/20 0.32
KCNH2 Q12809 4/20 0.32
ACHE P22303 1/20 0.31
MAPK13 O15264 1/20 0.31
RAF1 P04049 1/20 0.31
MAPK12 P53778 1/20 0.31
MAPK11 Q15759 1/20 0.31
MAPK14 Q16539 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5819870 0.90 MAPK14 (0.36) PTGDR2BRAFKMOMAPK13RAF1
SCHEMBL5818348 0.85 MAPK14 (0.36) PTGDR2MAPK13RAF1MAPK12MAPK11
SCHEMBL5819125 0.83 CKS1B (0.38) PTGDR2BRAF
SCHEMBL5819534 0.81 MAPK14 (0.38) MAPK13MAPK12MAPK11MAPK14
SCHEMBL5819457 0.80 EGFR (0.39) MAPK11MAPK14
SCHEMBL5818792 0.80 MAPK14 (0.40) KMOMAPK13MAPK12MAPK11MAPK14
SCHEMBL5818359 0.79 KCNH2 (0.41) BRAFKCNH2RAF1MAPK14
SCHEMBL5819170 0.78 CAMK2D (0.47) MAPK13RAF1MAPK12MAPK11MAPK14
SCHEMBL5815121 0.77 BRAF (0.50) BRAFKCNH2ACHERAF1MAPK14
SCHEMBL5814145 0.75 PIK3CA (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006137658-A1 NEW SUBSTITUTED 1,3-THIAZOLE DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF HAVING IMMUNOSUPPRESSION AND INFLAMMATION INHIBITORY ACITIVITY, INTERMEDIATE COMPOUNDS OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, A PROCESS FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DONGBU HITEK CO., LTD. (KR) 2006-12-28 WO disclosed