SCHEMBL5818784

SCHEMBL5818784

Cc1cccc(-c2nc(C3CCNCC3)sc2-c2n[c]ncc2C2CC2)c1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 3/20 0.45
GABRB2 P47870 3/20 0.45
HTR2C P28335 2/20 0.37
MAPK14 Q16539 2/20 0.37
KCNH2 Q12809 2/20 0.37
ACHE P22303 1/20 0.36
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
HTR7 P34969 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5819814 0.96 GABRA1 (0.44) GABRA1GABRB2HTR2CMAPK14KCNH2
SCHEMBL5819266 0.89 KCNH2 (0.39) GABRA1GABRB2KCNH2ACHE
SCHEMBL5814885 0.88 MAPK14 (0.40) GABRA1GABRB2MAPK14KCNH2CNR1
SCHEMBL5813729 0.86 MEN1 (0.42) HTR2CMAPK14MEN1KMT2A
SCHEMBL5814140 0.85 GABRA1 (0.39) GABRA1GABRB2HTR2CMAPK14KCNH2
SCHEMBL5813870 0.84 MAPK14 (0.39) GABRA1GABRB2MAPK14KCNH2
SCHEMBL5818833 0.83 MEN1 (0.41) HTR2CMAPK14MEN1KMT2A
SCHEMBL5815410 0.82 KCNH2 (0.47) KCNH2ACHE
SCHEMBL5812990 0.82 MEN1 (0.41) HTR2CMAPK14MEN1KMT2A
SCHEMBL5814697 0.82 MEN1 (0.38) HTR2CKCNH2ACHEMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006137658-A1 NEW SUBSTITUTED 1,3-THIAZOLE DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF HAVING IMMUNOSUPPRESSION AND INFLAMMATION INHIBITORY ACITIVITY, INTERMEDIATE COMPOUNDS OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, A PROCESS FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DONGBU HITEK CO., LTD. (KR) 2006-12-28 WO claimed