SCHEMBL5818970

SCHEMBL5818970

COc1ccc(-c2nc(C3CCN(C)CC3)sc2-c2ccnc([C@@](C)(N)c3ccccc3)n2)cc1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.47
RAF1 P04049 1/20 0.47
ERBB2 P04626 1/20 0.47
SRC P12931 1/20 0.47
KDR P35968 1/20 0.47
MAPK8 P45983 1/20 0.47
MAPK9 P45984 1/20 0.47
KCNH2 Q12809 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5819634 0.89 KCNH2 (0.48) KCNH2
SCHEMBL5819618 0.85 EGFR (0.43) EGFRRAF1ERBB2SRCKDR
SCHEMBL5818662 0.84 KCNH2 (0.44) EGFRRAF1ERBB2SRCKDR
SCHEMBL5819631 0.84 EGFR (0.44) EGFRRAF1ERBB2SRCKDR
SCHEMBL5816216 0.84 EGFR (0.48) EGFRRAF1ERBB2SRCKDR
SCHEMBL5814016 0.83 EGFR (0.43) EGFRRAF1ERBB2SRCKDR
SCHEMBL5823310 0.80 ALDH1A1 (0.51) KCNH2
SCHEMBL5818972 0.80 EGFR (0.64) EGFRRAF1ERBB2SRCKDR
SCHEMBL5815611 0.80 KCNH2 (0.54) EGFRRAF1ERBB2SRCKDR
SCHEMBL5820563 0.79 KMT2A (0.47) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006137658-A1 NEW SUBSTITUTED 1,3-THIAZOLE DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF HAVING IMMUNOSUPPRESSION AND INFLAMMATION INHIBITORY ACITIVITY, INTERMEDIATE COMPOUNDS OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, A PROCESS FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DONGBU HITEK CO., LTD. (KR) 2006-12-28 WO claimed