SCHEMBL5819799

SCHEMBL5819799

CNc1nc(-c2ccc(F)cc2)c(-c2ccnc([C@@](C)(N)c3ccccc3)n2)s1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 2/20 0.45
CDK9 P50750 2/20 0.45
EGFR P00533 6/20 0.45
TGFBR1 P36897 1/20 0.39
KCNH2 Q12809 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
BRAF P15056 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5813644 0.83 CCNT1 (0.47) CCNT1CDK9TGFBR1BRAF
SCHEMBL5817990 0.81 PTGDR2 (0.36) TGFBR1KCNH2
SCHEMBL5817615 0.78 KCNH2 (0.57) EGFRKCNH2
SCHEMBL5818629 0.78 KCNH2 (0.60) KCNH2
SCHEMBL30409799 0.78 EGFR (0.49) CCNT1CDK9EGFRTGFBR1KCNH2
SCHEMBL29039434 0.78 EGFR (0.49) CCNT1CDK9EGFRTGFBR1KCNH2
SCHEMBL5819806 0.77 MAPK13 (0.56) CCNT1CDK9EGFR
SCHEMBL5819805 0.77 MAPK13 (0.56) CCNT1CDK9EGFR
SCHEMBL5822178 0.73 EGFR (0.46) CCNT1CDK9EGFRTGFBR1KCNH2
SCHEMBL5819107 0.70 ADORA2A (0.38) KDM4EMAPTBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006137658-A1 NEW SUBSTITUTED 1,3-THIAZOLE DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF HAVING IMMUNOSUPPRESSION AND INFLAMMATION INHIBITORY ACITIVITY, INTERMEDIATE COMPOUNDS OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, A PROCESS FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DONGBU HITEK CO., LTD. (KR) 2006-12-28 WO disclosed