SCHEMBL5822178

SCHEMBL5822178

CNc1nc(-c2ccc(F)cc2)c(-c2ccnc([S+](C)[O-])n2)s1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.46
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
CCNT1 O60563 1/20 0.42
CDK9 P50750 1/20 0.42
KCNH2 Q12809 2/20 0.40
TGFBR1 P36897 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5819549 0.84 TGFBR1 (0.55) EGFRKDM4EALDH1A1MAPTKCNH2
SCHEMBL30409799 0.82 EGFR (0.49) EGFRKDM4EALDH1A1MAPTCCNT1
SCHEMBL29039434 0.82 EGFR (0.49) EGFRKDM4EALDH1A1MAPTCCNT1
SCHEMBL5822172 0.82 PTGS2 (0.41) EGFRKCNH2TGFBR1
SCHEMBL5818004 0.79 MEN1 (0.33) KCNH2TGFBR1
SCHEMBL5818469 0.78 KCNH2 (0.54) EGFRALDH1A1KCNH2
SCHEMBL5819408 0.76 KCNH2 (0.62) KCNH2
SCHEMBL5817608 0.74 CDK2 (0.43) EGFRALDH1A1MAPTKCNH2
SCHEMBL5819799 0.73 CCNT1 (0.45) EGFRKDM4EALDH1A1MAPTCCNT1
SCHEMBL5819806 0.72 MAPK13 (0.56) EGFRCCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006137658-A1 NEW SUBSTITUTED 1,3-THIAZOLE DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF HAVING IMMUNOSUPPRESSION AND INFLAMMATION INHIBITORY ACITIVITY, INTERMEDIATE COMPOUNDS OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, A PROCESS FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DONGBU HITEK CO., LTD. (KR) 2006-12-28 WO disclosed