SCHEMBL5820830

SCHEMBL5820830

CCOC(=O)CC(c1ccccc1)n1ccc2c(CCc3ccc4c(n3)N(C(=O)OC(C)(C)C)CCC4)cccc21

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 15/20 0.54
ITGAV P06756 15/20 0.54
ITGB5 P18084 6/20 0.54
L3MBTL1 Q9Y468 1/20 0.36
MCL1 Q07820 1/20 0.31
ALDH1A1 P00352 1/20 0.31
ATM Q13315 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5809683 0.86 ITGB3 (0.66) ITGB3ITGAVITGB5
SCHEMBL861676 0.83 ITGB3 (0.56) ITGB3ITGAVITGB5
SCHEMBL5815728 0.81 ITGB3 (0.81) ITGB3ITGAVITGB5
SCHEMBL861296 0.80 ITGB3 (0.58) ITGB3ITGAVITGB5
SCHEMBL861561 0.79 ITGB3 (0.52) ITGB3ITGAVITGB5
SCHEMBL861581 0.78 ITGB3 (0.58) ITGB3ITGAVITGB5
SCHEMBL860336 0.78 ITGB3 (0.59) ITGB3ITGAVITGB5
SCHEMBL861506 0.78 ITGB3 (0.51) ITGB3ITGAVITGB5
SCHEMBL862008 0.78 ITGB3 (0.57) ITGB3ITGAVITGB5
SCHEMBL860404 0.77 ITGB3 (0.57) ITGB3ITGAVITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006108040-A1 SUBSTITUTED INDOLES AND THEIR USE AS INTEGRIN ANTAGONISTS JANSSEN PHARMACEUTICA, N.V. (BE) 2006-10-12 WO disclosed
WO-2006072353-A1 AZETIDINE-SUBSTITUTED PYRAZOLINES AS PAR-1 ANTAGONISTS BAYER HEALTHCARE AG (DE) 2006-07-13 WO disclosed