SCHEMBL5821682

SCHEMBL5821682

CNc1c(C=Nc2cc([N+](=O)[O-])ccc2C)cnc2[nH]ccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
SMN1; SMN2 Q16637 2/20 0.44
NPC1 O15118 1/20 0.44
LMNA P02545 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
MAPT P10636 5/20 0.39
PKM P14618 1/20 0.39
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
TYK2 P29597 1/20 0.37
JAK3 P52333 1/20 0.37
TSHR P16473 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KDM4E B2RXH2 1/20 0.37
PIK3CA P42336 3/20 0.36
PIK3CD O00329 2/20 0.36
MAOA P21397 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5821680 1.00 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2NPC1LMNAMAPK1
SCHEMBL5823344 0.73 KAT2B (0.42) ALDH1A1LMNAHTTMAPTMEN1
SCHEMBL1134969 0.68 PRKCI (0.44) KMT2AJAK2JAK1TYK2JAK3
SCHEMBL22025941 0.66 ALDH1A1 (0.61) ALDH1A1SMN1; SMN2NPC1LMNAMAPK1
SCHEMBL15555902 0.66 FGFR1 (0.42) JAK2JAK1TYK2JAK3
SCHEMBL15555901 0.66 FGFR1 (0.42) JAK2JAK1TYK2JAK3
SCHEMBL26220089 0.66 PRKCI (0.61) JAK2JAK1JAK3AXLPRKCI
SCHEMBL18926217 0.65 PRKCI (0.44) JAK2JAK1JAK3AXLPRKCI
SCHEMBL11494910 0.64 ALDH1A1 (0.62) ALDH1A1SMN1; SMN2NPC1LMNAMAPK1
SCHEMBL17495401 0.62 PRKCI (0.46) ALDH1A1SMN1; SMN2NPC1MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006124731-A2 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2006-11-23 WO disclosed