SCHEMBL5821773

SCHEMBL5821773

CSc1nc(Nc2ccc(N3CCOCC3)cc2)cc(N2CCN(CC(=O)NCCN3CCOCC3)CC2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.45
AURKB Q96GD4 1/20 0.45
RET P07949 2/20 0.44
TSHR P16473 1/20 0.43
CYP1A2 P05177 1/20 0.43
MAPT P10636 2/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
ZAP70 P43403 1/20 0.41
IGF1R P08069 1/20 0.41
POLB P06746 1/20 0.41
RGS12 O14924 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDR P35968 4/20 0.40
BRAF P15056 2/20 0.40
RAF1 P04049 1/20 0.40
PDGFRB P09619 1/20 0.40
KIT P10721 1/20 0.40
FGFR1 P11362 1/20 0.40
TEK Q02763 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5820767 0.97 AURKA (0.43) AURKAAURKBRETTSHRCYP1A2
SCHEMBL5820626 0.96 AURKA (0.43) AURKAAURKBRETTSHRCYP1A2
SCHEMBL5823053 0.92 AURKA (0.45) AURKAAURKBRETCYP1A2MAPT
SCHEMBL5824056 0.91 AURKA (0.48) AURKAAURKBRETCYP1A2MAPT
SCHEMBL5815015 0.89 AURKA (0.47) AURKAAURKBRETCYP1A2MAPT
SCHEMBL5820813 0.88 NAMPT (0.47) AURKAAURKBRETCYP1A2MAPT
SCHEMBL5820773 0.88 AURKA (0.42) AURKAAURKBRETCYP1A2MAPT
SCHEMBL5402668 0.87 AURKA (0.48) AURKAAURKBCYP1A2MAPTTP53
SCHEMBL5823423 0.86 AURKA (0.46) AURKAAURKBRETCYP1A2MAPT
SCHEMBL5822050 0.84 INSR (0.46) AURKAAURKBCYP1A2MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006137706-A1 6-(4-SUBSTITUTED-ANILINO)PYRIMIDINE DERIVATIVES, METHOD FOR PREPARING THEREOF AND ANTIVIRAL PHARMACEUTICAL COMPOSITION COMPRISING THE SAME B & C BIOPHARM. CO., LTD. (KR) 2006-12-28 WO claimed
WO-2006137706-A1 6-(4-SUBSTITUTED-ANILINO)PYRIMIDINE DERIVATIVES, METHOD FOR PREPARING THEREOF AND ANTIVIRAL PHARMACEUTICAL COMPOSITION COMPRISING THE SAME B & C BIOPHARM. CO., LTD. (KR) 2006-12-28 WO disclosed