SCHEMBL5822073

SCHEMBL5822073

COc1ccccc1-c1nc2ccc(Oc3ccc(F)cc3)cc2c(=O)n1CC1CCCN(CC(C)C)C1

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 6/20 0.69
GHSR Q92847 14/20 0.68
KCNH2 Q12809 5/20 0.60
HTR2C P28335 1/20 0.49
CYP3A4 P08684 1/20 0.47
AVPR1B P47901 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21632610 0.83 GHSR (0.85) CYP2D6GHSRKCNH2HTR2CCYP3A4
SCHEMBL21632609 0.83 GHSR (0.85) CYP2D6GHSRKCNH2HTR2CCYP3A4
SCHEMBL5791022 0.82 GHSR (0.85) CYP2D6GHSRKCNH2HTR2CCYP3A4
SCHEMBL20528762 0.82 CYP2D6 (1.00) CYP2D6GHSRKCNH2CYP3A4
SCHEMBL20528764 0.82 CYP2D6 (1.00) CYP2D6GHSRKCNH2CYP3A4
SCHEMBL5823927 0.79 CYP2D6 (0.80) CYP2D6GHSRKCNH2HTR2CCYP3A4
SCHEMBL5794076 0.78 CYP2D6 (0.79) CYP2D6GHSRKCNH2HTR2CCYP3A4
SCHEMBL5794769 0.78 CYP2D6 (0.62) CYP2D6GHSRKCNH2HTR2CCYP3A4
SCHEMBL10064690 0.76 GHSR (1.00) CYP2D6GHSRKCNH2
SCHEMBL2742704 0.76 GHSR (1.00) CYP2D6GHSRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006012577-A2 QUINAZOLINONE DERIVATIVES USEFUL FOR THE REGULATION OF GLUCOSE HOMEOSTASIS AND FOOD INTAKE BAYER PHARMACEUTICALS CORPORATION (US) 2006-02-02 WO disclosed