SCHEMBL5794769

SCHEMBL5794769

CCN1CCCC(Cn2c(-c3ccccc3OC)nc3ccc(Br)cc3c2=O)C1

nearest known ligand 0.62

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.62
HTR2C P28335 1/20 0.62
GHSR Q92847 16/20 0.52
KCNH2 Q12809 6/20 0.48
CYP3A4 P08684 1/20 0.48
AVPR1B P47901 1/20 0.45
MAPK8 P45983 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5793472 0.88 GHSR (0.49) CYP2D6HTR2CGHSRKCNH2CYP3A4
SCHEMBL5792698 0.84 GHSR (0.48) CYP2D6HTR2CGHSRKCNH2CYP3A4
SCHEMBL5794299 0.81 CYP2D6 (0.57) CYP2D6HTR2CGHSRKCNH2CYP3A4
SCHEMBL5822073 0.78 CYP2D6 (0.69) CYP2D6HTR2CGHSRKCNH2CYP3A4
SCHEMBL5794926 0.77 CYP2D6 (0.69) CYP2D6HTR2CGHSRKCNH2CYP3A4
SCHEMBL5791441 0.77 GHSR (0.76) CYP2D6HTR2CGHSRKCNH2CYP3A4
SCHEMBL5794423 0.77 CYP2D6 (0.79) CYP2D6HTR2CGHSRKCNH2CYP3A4
SCHEMBL5805037 0.75 CYP2D6 (0.65) CYP2D6HTR2CGHSRKCNH2CYP3A4
SCHEMBL5792759 0.75 CYP2D6 (0.65) CYP2D6HTR2CGHSRKCNH2CYP3A4
SCHEMBL5792756 0.75 CYP2D6 (0.65) CYP2D6HTR2CGHSRKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006012577-A2 QUINAZOLINONE DERIVATIVES USEFUL FOR THE REGULATION OF GLUCOSE HOMEOSTASIS AND FOOD INTAKE BAYER PHARMACEUTICALS CORPORATION (US) 2006-02-02 WO disclosed