SCHEMBL582239

SCHEMBL582239

Oc1c(Br)cc(Cl)cc1Br.Oc1cc(Cl)ccc1Cl

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 6/20 0.68
HSD17B10 Q99714 6/20 0.68
ALDH1A1 P00352 4/20 0.68
CYP3A4 P08684 3/20 0.68
TDP1 Q9NUW8 2/20 0.68
AMY1A P0DUB6 2/20 0.45
ERN1 O75460 1/20 0.44
HPGD P15428 4/20 0.40
HSP90AA1 P07900 2/20 0.40
NR1I2 O75469 1/20 0.40
LMNA P02545 1/20 0.40
TTR P02766 1/20 0.40
PGR P06401 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
MAPT P10636 1/20 0.40
HSPA5 P11021 1/20 0.40
CBR1 P16152 1/20 0.40
TBXA2R P21731 1/20 0.40
SLC6A2 P23975 1/20 0.40
AGTR1 P30556 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19553825 0.82 HSD17B10 (1.00) TSHRHSD17B10ALDH1A1CYP3A4TDP1
SCHEMBL177878 0.82
SCHEMBL16824107 0.80 HSD17B10 (0.94) TSHRHSD17B10ALDH1A1CYP3A4TDP1
Potassium SCHEMBL31408933 0.80 HSD17B10 (0.94) TSHRHSD17B10ALDH1A1CYP3A4TDP1
Potassium SCHEMBL31408932 0.80 HSD17B10 (0.94) TSHRHSD17B10ALDH1A1CYP3A4TDP1
SCHEMBL27242086 0.80 HSD17B10 (0.94) TSHRHSD17B10ALDH1A1CYP3A4TDP1
Potassium SCHEMBL31408934 0.80 HSD17B10 (0.94) TSHRHSD17B10ALDH1A1CYP3A4TDP1
SCHEMBL7119646 0.80 ERN1 (0.60) TSHRHSD17B10ALDH1A1CYP3A4TDP1
SCHEMBL264625 0.78 ERN1 (0.54) TSHRHSD17B10ALDH1A1CYP3A4TDP1
SCHEMBL11209383 0.77 HSD17B10 (0.77) TSHRHSD17B10ALDH1A1CYP3A4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1543061-A1 METHOD OF PREPARING TRANSPARENT SILICONE-CONTAINING COPOLYCARBONATES GENERAL ELECTRIC COMPANY (US) 2005-06-22 EP claimed
US-6833422-B2 Interfacial polymerization of polycarbonates with polysiloxanes, then endcapping to form haze-free polycarbonatepolysiloxane copolymers GENERAL ELECTRIC COMPANY 2004-12-21 US claimed
WO-2004016674-A1 METHOD OF PREPARING TRANSPARENT SILICONE-CONTAINING COPOLYCARBONATES GENERAL ELECTRIC COMPANY (US) 2004-02-26 WO claimed
US-20040039145-A1 Method of preparing transparent silicone-containing copolycarbonates GENERAL ELECTRIC COMPANY 2004-02-26 US claimed
US-20020111456-A1 Method of polycarbonate preparation SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2002-08-15 US claimed
WO-2001085825-A2 METHOD OF POLYCARBONATE PREPARATION GENERAL ELECTRIC COMPANY (US) 2001-11-15 WO claimed
EP-1307499-B2 CONTINUOUS PREPARATION OF POLYCARBONATE GEN ELECTRIC (US) 2012-02-15 EP disclosed
EP-1307499-B1 CONTINUOUS PREPARATION OF POLYCARBONATE GEN ELECTRIC (US) 2006-10-25 EP disclosed
EP-1543061-B1 METHOD OF PREPARING TRANSPARENT SILICONE-CONTAINING COPOLYCARBONATES GEN ELECTRIC (US) 2006-08-30 EP disclosed
EP-1543061-A1 METHOD OF PREPARING TRANSPARENT SILICONE-CONTAINING COPOLYCARBONATES GENERAL ELECTRIC COMPANY (US) 2005-06-22 EP disclosed
US-6833422-B2 Interfacial polymerization of polycarbonates with polysiloxanes, then endcapping to form haze-free polycarbonatepolysiloxane copolymers GENERAL ELECTRIC COMPANY 2004-12-21 US disclosed
WO-2004016674-A1 METHOD OF PREPARING TRANSPARENT SILICONE-CONTAINING COPOLYCARBONATES GENERAL ELECTRIC COMPANY (US) 2004-02-26 WO disclosed
US-20040039145-A1 Method of preparing transparent silicone-containing copolycarbonates GENERAL ELECTRIC COMPANY 2004-02-26 US disclosed
US-6562937-B2 Endcapping with phenol GENERAL ELECTRIC COMPANY 2003-05-13 US disclosed
EP-1307499-A2 CONTINUOUS PREPARATION OF POLYCARBONATE GENERAL ELECTRIC COMPANY (US) 2003-05-07 EP disclosed
US-20020111456-A1 Method of polycarbonate preparation SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2002-08-15 US disclosed
US-20020035234-A1 Continuous preparation of polycarbonate GENERAL ELECTRIC COMPANY 2002-03-21 US disclosed
WO-2002008311-A2 CONTINUOUS PREPARATION OF POLYCARBONATE GENERAL ELECTRIC COMPANY (US) 2002-01-31 WO disclosed
WO-2001085825-A2 METHOD OF POLYCARBONATE PREPARATION GENERAL ELECTRIC COMPANY (US) 2001-11-15 WO disclosed