SCHEMBL5823772

SCHEMBL5823772

C[C@H]1c2cccn2-c2ccc(F)cc2N1C(=O)c1ccccc1O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 10/20 0.40
PDK2 Q15119 10/20 0.40
PDK3 Q15120 10/20 0.40
PDK4 Q16654 10/20 0.40
HSP90AA1 P07900 2/20 0.40
PTPN2 P17706 1/20 0.40
PTPN1 P18031 1/20 0.40
KCNMA1 Q12791 1/20 0.40
MAPT P10636 2/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 1/20 0.34
KLK7 P49862 1/20 0.34
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
ALOX12 P18054 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4491393 0.83 KMT2A (0.43) PDK1PDK2PDK3PDK4HSP90AA1
SCHEMBL4503272 0.83 KMT2A (0.43) PDK1PDK2PDK3PDK4HSP90AA1
SCHEMBL4501038 0.83 KMT2A (0.43) PDK1PDK2PDK3PDK4HSP90AA1
SCHEMBL4502357 0.81 KMT2A (0.39) PDK1PDK2PDK3PDK4HSP90AA1
SCHEMBL4489743 0.81 KMT2A (0.39) PDK1PDK2PDK3PDK4HSP90AA1
SCHEMBL4495844 0.81 KMT2A (0.39) PDK1PDK2PDK3PDK4HSP90AA1
SCHEMBL4503738 0.78 ALDH1A1 (0.44) PTPN1KDM4EALDH1A1MEN1NPC1
SCHEMBL4497604 0.76 ALDH1A1 (0.48) PTPN1KDM4EALDH1A1MEN1NPC1
SCHEMBL4498228 0.76 PDK1 (0.53) PDK1PDK2PDK3PDK4HSP90AA1
SCHEMBL4503844 0.75 PDK1 (0.48) PDK1PDK2PDK3PDK4HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006068928-A1 PYRROLO[1,2-A]QUINOXALIN-5-(4H)-YL)SULFONYLS AND CARBONYLS AND THEIR USE AS ESTROGENIC AGENTS WYETH (US) 2006-06-29 WO disclosed