SCHEMBL5828296

SCHEMBL5828296

COc1ccc2[nH]c(C=Cc3ccccc3Cl)cc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 5/20 0.55
RELA Q04206 1/20 0.55
KDM4E B2RXH2 2/20 0.49
MAPT P10636 2/20 0.49
ALDH1A1 P00352 1/20 0.49
ABCG2 Q9UNQ0 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
MAOB P27338 2/20 0.48
AXL P30530 1/20 0.48
FLT3 P36888 3/20 0.47
CASP3 P42574 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
PDGFRB P09619 2/20 0.45
PDGFRA P16234 2/20 0.45
CYP1A2 P05177 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5828295 1.00 NFE2L2 (0.55) NFE2L2RELAKDM4EMAPTALDH1A1
SCHEMBL5827969 0.89 AXL (0.50) NFE2L2RELAKDM4EMAPTALDH1A1
SCHEMBL5827972 0.89 AXL (0.50) NFE2L2RELAKDM4EMAPTALDH1A1
SCHEMBL5829136 0.89 AXL (0.50) NFE2L2RELAKDM4EMAPTALDH1A1
SCHEMBL5829134 0.89 AXL (0.50) NFE2L2RELAKDM4EMAPTALDH1A1
SCHEMBL5828046 0.85 FLT3 (0.51) KDM4EMAPTALDH1A1MEN1KMT2A
SCHEMBL5828048 0.85 FLT3 (0.51) KDM4EMAPTALDH1A1MEN1KMT2A
SCHEMBL5829021 0.84 MEN1 (0.49) KDM4EMAPTMEN1KMT2ANPC1
SCHEMBL5829018 0.84 MEN1 (0.49) KDM4EMAPTMEN1KMT2ANPC1
SCHEMBL5828840 0.83 CYP1A1 (0.46) NFE2L2KDM4EMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7094798-B1 Inhibitors of checkpoint kinases (Wee1 and Chk1) PFIZER INC (US) 2006-08-22 US disclosed
EP-1501831-A1 INHIBITORS OF CHECKPOINT KINASES (WEE1 AND CHK1) WARNER-LAMBERT COMPANY LLC (US) 2005-02-02 EP disclosed
WO-2003091255-A1 INHIBITORS OF CHECKPOINT KINASES (WEE1 AND CHK1) WARNER-LAMBERT COMPANY LLC (US) 2003-11-06 WO disclosed