SCHEMBL5828319

SCHEMBL5828319

COc1cc2cc(C=O)[nH]c2cc1OCc1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 2/20 0.67
SRD5A2 P31213 2/20 0.67
CTSV O60911 2/20 0.54
CTSL P07711 2/20 0.54
RXFP1 Q9HBX9 1/20 0.48
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
PDGFRB P09619 1/20 0.44
PDGFRA P16234 1/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MAPT P10636 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ERN1 O75460 1/20 0.44
HPGD P15428 1/20 0.43
CYP2A6 P11509 1/20 0.43
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5829207 0.86 SRD5A1 (0.62) SRD5A1SRD5A2CTSVCTSLRXFP1
SCHEMBL5829277 0.86 SRD5A1 (0.62) SRD5A1SRD5A2CTSVCTSLRXFP1
SCHEMBL5829209 0.86 SRD5A1 (0.62) SRD5A1SRD5A2CTSVCTSLRXFP1
SCHEMBL13946720 0.82 EHMT2 (0.55) SRD5A1SRD5A2RXFP1KMT2AMEN1
SCHEMBL7169748 0.80 SRD5A2 (1.00) SRD5A1SRD5A2CTSVCTSLRXFP1
SCHEMBL3243291 0.80 SRD5A2 (1.00) SRD5A1SRD5A2CTSVCTSLRXFP1
SCHEMBL28820805 0.80 SRD5A1 (0.66) SRD5A1SRD5A2CTSVCTSLRXFP1
SCHEMBL30997265 0.80 SRD5A1 (0.66) SRD5A1SRD5A2CTSVCTSLRXFP1
SCHEMBL5829229 0.78 SRD5A2 (0.82) SRD5A1SRD5A2CTSVCTSLRXFP1
SCHEMBL7159304 0.78 SRD5A2 (0.82) SRD5A1SRD5A2CTSVCTSLRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7094798-B1 Inhibitors of checkpoint kinases (Wee1 and Chk1) PFIZER INC (US) 2006-08-22 US disclosed
EP-1501831-A1 INHIBITORS OF CHECKPOINT KINASES (WEE1 AND CHK1) WARNER-LAMBERT COMPANY LLC (US) 2005-02-02 EP disclosed
WO-2003091255-A1 INHIBITORS OF CHECKPOINT KINASES (WEE1 AND CHK1) WARNER-LAMBERT COMPANY LLC (US) 2003-11-06 WO disclosed