SCHEMBL5828446

SCHEMBL5828446

COc1cc(Br)c2oc(C=O)cc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 6/20 0.47
MAOA P21397 2/20 0.47
CYP2A6 P11509 2/20 0.40
F2RL3 Q96RI0 2/20 0.40
SLC22A12 Q96S37 1/20 0.38
ALDH1A1 P00352 2/20 0.36
TP53 P04637 2/20 0.36
HPGD P15428 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MAPT P10636 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PRKDC P78527 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP1A1 P04798 1/20 0.34
CYP1B1 Q16678 1/20 0.34
ERN1 O75460 2/20 0.34
ADORA3 P0DMS8 1/20 0.33
APP P05067 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL120165 0.83 ERN1 (0.44) MAOBCYP2A6ALDH1A1TP53HPGD
SCHEMBL5746295 0.76 SLC22A12 (0.46) MAOBMAOACYP2A6F2RL3SLC22A12
SCHEMBL13202363 0.75 MAOB (0.51) MAOBMAOAF2RL3SLC22A12ALDH1A1
SCHEMBL5828926 0.73 NFE2L2 (0.49) MAOBMAOAALDH1A1TP53HPGD
SCHEMBL5828924 0.73 NFE2L2 (0.49) MAOBMAOAALDH1A1TP53HPGD
SCHEMBL11746052 0.72 PIM1 (0.61) MAOBMAOAF2RL3SLC22A12ALDH1A1
SCHEMBL4130113 0.72 LMNA (0.51) MAOBMAOAF2RL3SLC22A12ALDH1A1
SCHEMBL29985195 0.71 APP (0.60) MAOBCYP2A6ALDH1A1HPGDAPP
SCHEMBL120294 0.71 APP (0.60) MAOBCYP2A6ALDH1A1HPGDAPP
SCHEMBL5829219 0.71 PIM1 (0.46) MAOBMAOAF2RL3SLC22A12ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7094798-B1 Inhibitors of checkpoint kinases (Wee1 and Chk1) PFIZER INC (US) 2006-08-22 US disclosed
EP-1501831-A1 INHIBITORS OF CHECKPOINT KINASES (WEE1 AND CHK1) WARNER-LAMBERT COMPANY LLC (US) 2005-02-02 EP disclosed
WO-2003091255-A1 INHIBITORS OF CHECKPOINT KINASES (WEE1 AND CHK1) WARNER-LAMBERT COMPANY LLC (US) 2003-11-06 WO disclosed