SCHEMBL5831475

SCHEMBL5831475

CCCc1ccc(S(=O)(=O)Nc2nnc(CC(=O)N(CC)CC)s2)cc1

nearest known ligand 0.67

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 9/20 0.67
GAB1 Q13480 4/20 0.67
IRS1 P35568 3/20 0.67
PKM P14618 2/20 0.55
ALDH1A1 P00352 1/20 0.55
HSD17B10 Q99714 1/20 0.50
ATM Q13315 1/20 0.49
RECQL P46063 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5830619 0.90 AKT1 (0.63) AKT1GAB1IRS1PKMALDH1A1
SCHEMBL5831043 0.88 AKT1 (0.63) AKT1GAB1IRS1PKMALDH1A1
SCHEMBL5832093 0.85 ATM (0.58) AKT1GAB1IRS1PKMALDH1A1
SCHEMBL3251192 0.82 AKT1 (0.48) AKT1GAB1IRS1ALDH1A1
SCHEMBL5832128 0.81 AKT1 (0.47) AKT1GAB1IRS1ALDH1A1
SCHEMBL283045 0.80 AKT1 (1.00) AKT1GAB1IRS1
SCHEMBL3605393 0.80 HSD17B1 (0.59) AKT1GAB1IRS1PKMALDH1A1
SCHEMBL5831319 0.79 AKT1 (0.60) AKT1GAB1IRS1PKMALDH1A1
SCHEMBL282664 0.79 AKT1 (1.00) AKT1GAB1IRS1
SCHEMBL5831265 0.79 AKT1 (0.59) AKT1GAB1IRS1PKMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1461327-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2004-09-29 EP claimed
US-20030130258-A1 Antidiabetic agents; liver disorders; cardiovascular disorders; dietetics BIOVITRUM AB (SE) 2003-07-10 US claimed
WO-2003044000-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2003-05-30 WO claimed
US-7074788-B2 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB (SE) 2006-07-11 US disclosed
EP-1461327-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2004-09-29 EP disclosed
US-20030130258-A1 Antidiabetic agents; liver disorders; cardiovascular disorders; dietetics BIOVITRUM AB (SE) 2003-07-10 US disclosed
WO-2003044000-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2003-05-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030130258-A1 Antidiabetic agents; liver disorders; cardiovascular disorders; dietetics CPT1A, HSD11B1, CES1 AKT1 2974/4885GAB1 2088/4885IRS1 51/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.