SCHEMBL5833007

SCHEMBL5833007

CC(C)(C)NC(=O)[C@H](Cc1ccc(OCc2ccccc2)cc1)NC(=O)[C@@H](N)Cc1ccncc1.CC(C)CCN[C@@H](Cc1ccncc1)C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IL1RN P18510 1/20 0.46
ERAP2 Q6P179 1/20 0.46
ERAP1 Q9NZ08 1/20 0.46
MME P08473 2/20 0.46
ACE P12821 2/20 0.46
CPA1 P15085 2/20 0.46
ACE2 Q9BYF1 2/20 0.46
PLG P00747 1/20 0.46
REN P00797 1/20 0.45
CTSL P07711 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
MMP9 P14780 1/20 0.43
MMP8 P22894 1/20 0.43
YAP1 P46937 1/20 0.42
PSMB1 P20618 2/20 0.42
PSMB9 P28065 2/20 0.42
PSMB5 P28074 2/20 0.42
PSMB10 P40306 2/20 0.42
PSMB2 P49721 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5833138 0.95 MME (0.50) IL1RNERAP2ERAP1MMEACE
SCHEMBL5833134 0.95 MME (0.50) IL1RNERAP2ERAP1MMEACE
SCHEMBL5833946 0.91 MME (0.52) ERAP2MMEACECPA1ACE2
SCHEMBL5833943 0.91 MME (0.52) ERAP2MMEACECPA1ACE2
SCHEMBL5833543 0.88 GPR132 (0.50) IL1RNERAP2ERAP1MMEACE
SCHEMBL5833547 0.88 GPR132 (0.50) IL1RNERAP2ERAP1MMEACE
SCHEMBL5832907 0.88 ACACB (0.49) MMEACECPA1ACE2PLG
SCHEMBL7440242 0.86 MME (0.53) IL1RNERAP2ERAP1MMEACE
SCHEMBL7440228 0.86 MME (0.53) IL1RNERAP2ERAP1MMEACE
SCHEMBL5833486 0.86 MAOB (0.44) MMEACECPA1ACE2PLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6989448-B2 Heteroaryl alkyl alpha substituted peptidylamine calcium channel blockers HU LAIN-YEN 2006-01-24 US disclosed
US-6166052-A Heteroaryl alkyl alpha substituted peptidylamine calcium channel blockers WARNER-LAMBERT COMPANY (US) 2000-12-26 US disclosed