SCHEMBL5833712

SCHEMBL5833712

CCc1cnc(-c2ccc(C(F)(F)F)cc2)[nH]c1=O

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
COMT P21964 1/20 0.65
SCN2A Q99250 2/20 0.51
TRPV1 Q8NER1 1/20 0.50
TNKS2 Q9H2K2 10/20 0.48
TNKS O95271 9/20 0.48
WNT3A P56704 6/20 0.48
PARP2 Q9UGN5 5/20 0.47
PARP1 P09874 5/20 0.46
KDM4E B2RXH2 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
RAB9A P51151 1/20 0.44
NPY5R Q15761 1/20 0.44
PARP14 Q460N5 1/20 0.42
PARP4 Q9UKK3 1/20 0.42
AXIN2 Q9Y2T1 1/20 0.42
PARP3 Q9Y6F1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11932719 0.80 SCN2A (0.47) COMTSCN2ATNKS2TNKSWNT3A
SCHEMBL2433653 0.79 COMT (1.00) COMTSCN2ATRPV1TNKS2TNKS
SCHEMBL7012072 0.78 RECQL (0.67) COMTSCN2ATRPV1TNKS2TNKS
SCHEMBL4376727 0.77 KDM4E (0.76) COMTKDM4EL3MBTL1RAB9A
SCHEMBL3586816 0.75 COMT (0.68) COMTSCN2ATRPV1TNKS2TNKS
SCHEMBL23736196 0.74 SCN2A (0.59) COMTSCN2ATRPV1TNKS2TNKS
SCHEMBL15331905 0.71 COMT (0.57) COMTSCN2ATRPV1TNKS2TNKS
SCHEMBL26202011 0.71 SCN2A (0.55) COMTSCN2ATRPV1TNKS2TNKS
SCHEMBL15693156 0.68 TNKS2 (0.54) COMTTNKS2TNKSWNT3APARP2
SCHEMBL25833757 0.68 SCN2A (0.55) SCN2ATRPV1NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7153861-B2 For therapy of atheroscelerosis SMITHKLINE BEECHAM P.L.C. (GB) 2006-12-26 US disclosed