SCHEMBL5836022

SCHEMBL5836022

O=C(CCCNC(=O)OCc1ccccc1)Nc1ncc(Br)s1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 1/20 0.60
CDK2 P24941 1/20 0.60
CDK5 Q00535 1/20 0.60
HTT P42858 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.55
MAPK10 P53779 1/20 0.55
SETD1B Q9UPS6 1/20 0.48
LMNA P02545 1/20 0.47
TGM2 P21980 1/20 0.46
MAPK1 P28482 2/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
TP53 P04637 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HSD17B10 Q99714 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5835710 0.85 CCNE1 (0.61) CCNE1CDK2CDK5HTTSMN1; SMN2
SCHEMBL5956259 0.84 CCNE1 (0.67) CCNE1CDK2CDK5HTTSMN1; SMN2
SCHEMBL5835640 0.82 CCNE1 (0.59) CCNE1CDK2CDK5HTTSMN1; SMN2
SCHEMBL5836908 0.81 CCNE1 (0.55) CCNE1CDK2CDK5HTTSMN1; SMN2
SCHEMBL5835981 0.80 HTT (0.48) CCNE1CDK2CDK5HTTSMN1; SMN2
SCHEMBL21533445 0.78 SETD1B (0.65) CCNE1CDK2CDK5SMN1; SMN2MAPK10
SCHEMBL32681311 0.76 HTT (0.71) HTTSMN1; SMN2LMNATGM2HDAC3
SCHEMBL5835922 0.76 CCNE1 (1.00) CCNE1CDK2CDK5HTTSMN1; SMN2
SCHEMBL8704472 0.76 MMP3 (0.60) HTTSMN1; SMN2LMNATGM2ALDH1A1
SCHEMBL8709704 0.75 MMP3 (0.59) HTTSMN1; SMN2LMNATGM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037929-B1 2-amino-thiazole derivatives, process for their preparation, and their use as antitumor agents PHARMACIA & UPJOHN S.P.A. (IT) 2006-05-02 US disclosed