SCHEMBL5838566

SCHEMBL5838566

COc1cc(O)c(C(=O)C=Cc2cc(OCc3ccccc3)c(OCc3ccccc3)c(OCc3ccccc3)c2)c(OC)c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.70
KMT2A Q03164 4/20 0.70
CYP3A4 P08684 3/20 0.70
TP53 P04637 2/20 0.70
ATM Q13315 1/20 0.70
HSD17B10 Q99714 1/20 0.70
ABCG2 Q9UNQ0 6/20 0.64
MEN1 O00255 3/20 0.62
KDM4E B2RXH2 2/20 0.62
HPGD P15428 2/20 0.62
TDP1 Q9NUW8 2/20 0.62
MCL1 Q07820 1/20 0.62
NFKB1 P19838 1/20 0.61
DPP4 P27487 1/20 0.61
NFKB2 Q00653 1/20 0.61
RELA Q04206 1/20 0.61
APP P05067 1/20 0.61
MKNK2 Q9HBH9 1/20 0.60
MAOA P21397 2/20 0.59
MAOB P27338 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5838556 1.00 MAPT (0.70) MAPTKMT2ACYP3A4TP53ATM
SCHEMBL30141094 0.93 PDE4A (0.63) MAPTKMT2ACYP3A4TP53ATM
SCHEMBL30892448 0.93 PDE4A (0.63) MAPTKMT2ACYP3A4TP53ATM
SCHEMBL24983864 0.93 PDE4A (0.63) MAPTKMT2ACYP3A4TP53ATM
SCHEMBL29179321 0.93 PDE4A (0.63) MAPTKMT2ACYP3A4TP53ATM
SCHEMBL5433412 0.90 ABCG2 (0.76) MAPTKMT2ACYP3A4TP53ATM
SCHEMBL30384422 0.90 ABCG2 (0.76) MAPTKMT2ACYP3A4TP53ATM
SCHEMBL25192256 0.90 ABCG2 (0.76) MAPTKMT2ACYP3A4TP53ATM
SCHEMBL25193887 0.90 ABCG2 (0.76) MAPTKMT2ACYP3A4TP53ATM
SCHEMBL30383596 0.90 ABCG2 (0.76) MAPTKMT2ACYP3A4TP53ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7122573-B2 Analogs of green tea polyphenols as chemotherapeutic and chemopreventive agents SRI INTERNATIONAL (US) 2006-10-17 US disclosed
US-7109236-B2 Analogs of green tea polyphenols as chemotherapeutic and chemopreventive agents SRI INTERNATIONAL (US) 2006-09-19 US disclosed
EP-1581512-A2 ANALOGS OF GREEN TEA POLYPHENOLS AS CHEMOTHERAPEUTIC AND CHEMOPREVENTIVE AGENTS SRI INTERNATIONAL (US) 2005-10-05 EP disclosed
US-20040192723-A1 Analogs of green tea polyphenols as chemotherapeutic and chemopreventive agents SRI INTERNATIONAL 2004-09-30 US disclosed
WO-2004052873-A9 ANALOGS OF GREEN TEA POLYPHENOLS AS CHEMOTHERAPEUTIC AND CHEMOPREVENTIVE AGENTS STANFORD RES INST INT (US) 2004-08-12 WO disclosed
WO-2004052873-A2 ANALOGS OF GREEN TEA POLYPHENOLS AS CHEMOTHERAPEUTIC AND CHEMOPREVENTIVE AGENTS SRI INTERNATIONAL (US) 2004-06-24 WO disclosed
US-20040110790-A1 Analogs of green tea polyphenols as chemotherapeutic and chemopreventive agents SRI INTERNATIONAL 2004-06-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040192723-A1 Analogs of green tea polyphenols as chemotherapeutic and chemopreventive agents TEAD4, TEAD3, TEAD1 MAPT 2442/4885KMT2A 2705/4885CYP3A4 121/4885
US-20040110790-A1 Analogs of green tea polyphenols as chemotherapeutic and chemopreventive agents TEAD4, TEAD3, TEAD1 MAPT 2442/4885KMT2A 2705/4885CYP3A4 121/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.